SCHEMBL31387927

SCHEMBL31387927

Nc1ncc(Br)nc1C(=O)Nc1ccncc1

nearest known ligand 0.76

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ATR Q13535 11/20 0.76
PRKCI P41743 4/20 0.66
GRM5 P41594 1/20 0.63
PRKDC P78527 2/20 0.62
CYP3A4 P08684 1/20 0.54
TBK1 Q9UHD2 4/20 0.51
IKBKE Q14164 3/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14059993 1.00 ATR (0.76) ATRPRKCIGRM5PRKDCCYP3A4
SCHEMBL559881 0.87 ATR (1.00) ATRGRM5PRKDCCYP3A4
SCHEMBL15724439 0.86 ATR (0.68) ATRPRKCIGRM5PRKDCCYP3A4
SCHEMBL411951 0.85 ATR (0.75) ATRPRKCIGRM5PRKDCCYP3A4
SCHEMBL1586135 0.84 ATR (0.74) ATRPRKCIGRM5PRKDCCYP3A4
SCHEMBL14136995 0.82 ATR (0.52) ATRPRKCIGRM5PRKDCCYP3A4
SCHEMBL1800565 0.81 ATR (0.58) ATRPRKCIGRM5PRKDCCYP3A4
SCHEMBL25346973 0.81 PRKCI (0.55) ATRPRKCIPRKDC
SCHEMBL19101125 0.80 ATR (0.90) ATRPRKDCCYP3A4
SCHEMBL31388033 0.79 ATR (0.68) ATRPRKCIGRM5PRKDCCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114341127-B Aminopyrazine compounds as HPK1 inhibitors and uses thereof 百济神州有限公司 2024-12-17 CN disclosed