SCHEMBL14156271

SCHEMBL14156271

CCOC(=O)C(NC(=O)OC(C)(C)C)c1csc(NC=O)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.43
SMN1; SMN2 Q16637 4/20 0.40
GAA P10253 2/20 0.40
PTPRB P23467 3/20 0.39
CYP1A2 P05177 3/20 0.37
CYP2C19 P33261 3/20 0.37
CYP2C9 P11712 2/20 0.37
HTT P42858 1/20 0.37
CTSK P43235 3/20 0.36
CTSS P25774 1/20 0.36
ALDH1A1 P00352 4/20 0.36
MAPT P10636 3/20 0.36
LMNA P02545 2/20 0.35
CYP3A4 P08684 1/20 0.35
TSHR P16473 1/20 0.35
PI4KB Q9UBF8 1/20 0.35
KCNH2 Q12809 1/20 0.35
KDM4E B2RXH2 1/20 0.34
PKM P14618 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9651601 0.91 ABCB1 (0.38) ABCB1SMN1; SMN2GAAPTPRBCYP1A2
Hydrochloric Acid SCHEMBL9653115 0.90 ABCB1 (0.38) ABCB1SMN1; SMN2GAAPTPRBCYP1A2
SCHEMBL22017474 0.87 SMN1; SMN2 (0.46) ABCB1SMN1; SMN2GAAPTPRBCYP1A2
SCHEMBL8868383 0.86 CTSK (0.39) ABCB1PTPRBCTSKCTSSPI4KB
SCHEMBL9652891 0.85 SMN1; SMN2 (0.41) ABCB1SMN1; SMN2GAAPTPRBCYP1A2
SCHEMBL7535850 0.83 TSHR (0.47) SMN1; SMN2GAACYP1A2CYP2C19CYP2C9
SCHEMBL9076717 0.83 ABCB1 (0.45) ABCB1SMN1; SMN2GAAPTPRBCYP1A2
SCHEMBL9074827 0.83 CYP1A2 (0.42) ABCB1SMN1; SMN2GAAPTPRBCYP1A2
SCHEMBL9652877 0.81 SMN1; SMN2 (0.37) ABCB1SMN1; SMN2GAAPTPRBCYP1A2
SCHEMBL9076896 0.81 ABCB1 (0.41) ABCB1SMN1; SMN2GAAPTPRBCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7381734-B2 Serine protease inhibitors TULARIK LIMITED (GB) 2008-06-03 US disclosed
US-7157585-B2 Serine protease inhibitors TULARIK LIMITED (GB) 2007-01-02 US disclosed