SCHEMBL14156604

SCHEMBL14156604

NC1=Nc2cc(F)ccc2Nc2ccc(C(F)(F)F)cc21

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 5/20 0.42
HRH1 P35367 1/20 0.42
PAK1 Q13153 1/20 0.42
TP53 P04637 2/20 0.37
MPL P40238 2/20 0.36
DRD2 P14416 4/20 0.35
BACE1 P56817 1/20 0.35
DRD1 P21728 2/20 0.34
HTR5A P47898 1/20 0.33
ALK Q9UM73 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4836832 0.99 CHRM1 (0.41) CHRM1HRH1PAK1TP53MPL
SCHEMBL14156596 0.90 TP53 (0.41) CHRM1HRH1PAK1TP53MPL
Hydrochloric Acid SCHEMBL4837164 0.89 TP53 (0.40) CHRM1HRH1PAK1TP53MPL
SCHEMBL14156601 0.86 MPL (0.39) CHRM1MPLBACE1
SCHEMBL14156616 0.85 DRD2 (0.40) CHRM1HRH1MPLDRD2DRD1
Hydrochloric Acid SCHEMBL4845753 0.85 MPL (0.38) CHRM1MPLBACE1
SCHEMBL4842627 0.84 TP53 (0.43) CHRM1TP53DRD2BACE1MAPT
Hydrochloric Acid SCHEMBL4837078 0.84 DRD2 (0.39) CHRM1HRH1MPLDRD2DRD1
Hydrochloric Acid SCHEMBL4835541 0.83 TP53 (0.42) CHRM1TP53DRD2BACE1MAPT
SCHEMBL14156619 0.80 DRD2 (0.49) CHRM1HRH1PAK1DRD2DRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7384934-B2 Piperazine substituted aryl benzodiazepines ELI LILLY AND COMPANY (US) 2008-06-10 US disclosed
US-7214673-B2 For therapy of psychosis and bipolar disorder ELI LILLY AND COMPANY (US) 2007-05-08 US disclosed