SCHEMBL14156702

SCHEMBL14156702

COCC[C@H]1CN(C2=Nc3cc(Cl)ccc3Nc3ccc(C)cc32)CCN1C

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 10/20 0.51
DRD1 P21728 8/20 0.51
CHRM1 P11229 5/20 0.51
DRD3 P35462 4/20 0.51
KCNH2 Q12809 4/20 0.51
DRD4 P21917 4/20 0.51
HRH1 P35367 3/20 0.51
HTR2A P28223 2/20 0.51
HRH4 Q9H3N8 2/20 0.51
CYP1A2 P05177 2/20 0.51
CHRM2 P08172 2/20 0.51
CHRM4 P08173 2/20 0.51
CYP3A4 P08684 2/20 0.51
CHRM5 P08912 2/20 0.51
CYP2D6 P10635 2/20 0.51
CHRM3 P20309 2/20 0.51
DRD5 P21918 2/20 0.51
HRH3 Q9Y5N1 2/20 0.51
NFKB1 P19838 2/20 0.51
BLM P54132 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6208004 1.00 DRD2 (0.51) DRD2DRD1CHRM1DRD3KCNH2
Succinic Acid SCHEMBL4848019 0.93 DRD2 (0.46) DRD2DRD1CHRM1DRD3KCNH2
Succinic Acid SCHEMBL4848015 0.93 DRD2 (0.46) DRD2DRD1CHRM1DRD3KCNH2
SCHEMBL14156704 0.89 CHRM1 (0.56) DRD2DRD1CHRM1KCNH2DRD4
SCHEMBL4844343 0.89 CHRM1 (0.53) DRD2DRD1CHRM1DRD3KCNH2
SCHEMBL4844352 0.89 CHRM1 (0.53) DRD2DRD1CHRM1DRD3KCNH2
SCHEMBL4844331 0.89 CHRM1 (0.53) DRD2DRD1CHRM1DRD3KCNH2
SCHEMBL14156705 0.88 DRD2 (0.48) DRD2DRD1CHRM1DRD3KCNH2
SCHEMBL14156716 0.88 DRD2 (0.65) DRD2DRD1CHRM1DRD3KCNH2
SCHEMBL14156715 0.88 DRD2 (0.51) DRD2DRD1CHRM1DRD3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7384934-B2 Piperazine substituted aryl benzodiazepines ELI LILLY AND COMPANY (US) 2008-06-10 US disclosed
US-7384934-B2 Piperazine substituted aryl benzodiazepines ELI LILLY AND COMPANY (US) 2008-06-10 US disclosed