SCHEMBL14176734

SCHEMBL14176734

CC1(C)OC2(C=C(C(=O)O)C(S(=O)(=O)Nc3ccc(F)cc3Cl)CC2)OC1(C)C

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR4 O00206 5/20 0.51
KMT2A Q03164 2/20 0.38
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
LMNA P02545 2/20 0.36
TP53 P04637 1/20 0.36
MAPT P10636 2/20 0.34
MEN1 O00255 1/20 0.34
NPY1R P25929 1/20 0.34
NPY2R P49146 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
POLB P06746 1/20 0.33
MRGPRX1 Q96LB2 1/20 0.33
ACLY P53396 1/20 0.33
NAMPT P43490 1/20 0.33
HTT P42858 1/20 0.33
HPGD P15428 1/20 0.32
PIK3CD O00329 1/20 0.32
PIK3CA P42336 1/20 0.32
PIK3CB P42338 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1865788 0.88 TLR4 (0.50) TLR4KMT2ANPC1RAB9ALMNA
SCHEMBL1866600 0.87 TLR4 (0.67) TLR4KMT2ALMNATP53NPSR1
SCHEMBL27592447 0.87 TLR4 (0.55) TLR4KMT2ANPC1RAB9ALMNA
SCHEMBL14176725 0.86 TLR4 (0.49) TLR4KMT2ANPC1RAB9ALMNA
SCHEMBL4138878 0.85 TLR4 (0.48) TLR4KMT2ANPC1RAB9ALMNA
SCHEMBL4146514 0.85 TLR4 (0.49) TLR4KMT2ANPC1RAB9ALMNA
SCHEMBL14136690 0.85 TLR4 (0.49) TLR4KMT2ANPC1RAB9ALMNA
SCHEMBL4141115 0.85 TLR4 (0.49) TLR4KMT2ANPC1RAB9ALMNA
SCHEMBL17727727 0.85 TLR4 (0.49) TLR4KMT2ANPC1RAB9ALMNA
SCHEMBL4144992 0.85 TLR4 (0.46) TLR4KMT2ANPC1RAB9ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1935879-A1 SUBSTITUTED CYCLOALKENE DERIVATIVE Daiichi Sankyo Company, Limited (JP) 2008-06-25 EP disclosed