SCHEMBL14178917

SCHEMBL14178917

CCOc1ccc(-n2c([C@H](N)CNC(=O)OC(C)(C)C)nc3c(c2=O)CCCN3)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA2D1 P54289 1/20 0.36
KMT2A Q03164 4/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
MAPK1 P28482 1/20 0.35
TP53 P04637 3/20 0.34
ALDH1A1 P00352 5/20 0.34
TSHR P16473 3/20 0.34
THRB P10828 2/20 0.34
HTT P42858 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
HPGD P15428 1/20 0.34
CYP2C19 P33261 1/20 0.34
MEN1 O00255 3/20 0.33
MAPT P10636 2/20 0.33
KDM4E B2RXH2 1/20 0.33
GLA P06280 1/20 0.33
GAA P10253 1/20 0.33
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4814189 0.86 TP53 (0.38) CACNA2D1KMT2ASMN1; SMN2MAPK1TP53
SCHEMBL14178889 0.86 TP53 (0.38) CACNA2D1KMT2ASMN1; SMN2MAPK1TP53
SCHEMBL14178918 0.83 CYP3A4 (0.40) KMT2ASMN1; SMN2MAPK1ALDH1A1CYP2C9
SCHEMBL1892286 0.78 MAPT (0.48) KMT2AMAPK1ALDH1A1MEN1MAPT
SCHEMBL1892283 0.78 MAPT (0.48) KMT2AMAPK1ALDH1A1MEN1MAPT
SCHEMBL14178925 0.76 CXCR3 (0.51) CXCR3
SCHEMBL14178931 0.75 CXCR3 (0.59) CXCR3
SCHEMBL4810109 0.72 TP53 (0.41) KMT2ASMN1; SMN2MAPK1TP53ALDH1A1
SCHEMBL4810832 0.70 CXCR3 (0.41) KMT2ASMN1; SMN2MAPK1TP53ALDH1A1
SCHEMBL4810840 0.70 CXCR3 (0.41) KMT2ASMN1; SMN2MAPK1TP53ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7375102-B2 Tetrahydroquinazolin-4(3H)-one-related and tetrahydropyrido[2,3-D]pyrimidin-4(3H)-one-related compounds, compositions and methods for their use AMGEN SF, LLC (US) 2008-05-20 US disclosed