SCHEMBL1418151

SCHEMBL1418151

CCOC(=O)CN(CC=CC(=O)Nc1ccc2ncnc(Nc3cccc(Br)c3)c2c1)CC(=O)OCC

nearest known ligand 0.80

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
EGFR P00533 20/20 0.80
ERBB2 P04626 12/20 0.80

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1418149 1.00 EGFR (0.80) EGFRERBB2
SCHEMBL1418144 0.94 EGFR (0.79) EGFRERBB2
SCHEMBL1418142 0.94 EGFR (0.79) EGFRERBB2
SCHEMBL6585840 0.89 EGFR (1.00) EGFRERBB2
SCHEMBL30115294 0.89 EGFR (1.00) EGFRERBB2
SCHEMBL867890 0.86 EGFR (1.00) EGFRERBB2
SCHEMBL867889 0.86 EGFR (1.00) EGFRERBB2
SCHEMBL30115339 0.86 EGFR (1.00) EGFRERBB2
SCHEMBL7208199 0.85 EGFR (1.00) EGFRERBB2
SCHEMBL2990560 0.85 EGFR (1.00) EGFRERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2298746-A1 4-amino- quinazoline and quinoline derivatives having an inhibitory effect on signal transduction mediated by tyrosine kinases Boehringer Ingelheim Pharma GmbH & Co. KG (DE) 2011-03-23 EP disclosed
US-6972288-B1 4-amino-quinazoline and quinoline derivatives having an inhibitory effect on signal transduction mediated by tyrosine kinases BOEHRINGER INGELHEIM PHARMA KG (DE) 2005-12-06 US disclosed