SCHEMBL14185482

SCHEMBL14185482

Cc1cc(N)c(C=N)cc1I

nearest known ligand 0.36

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.36
CYP3A4 P08684 1/20 0.36
TSHR P16473 1/20 0.36
CD44 P16070 1/20 0.32
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20439331 0.92 CYP3A4 (0.31) MAPK1CYP3A4TSHR
SCHEMBL20109373 0.82 CYP3A4 (0.48) MAPK1CYP3A4TSHRCD44ALDH1A1
SCHEMBL19535201 0.80 CYP3A4 (0.52) MAPK1CYP3A4TSHRCD44ALDH1A1
SCHEMBL12181242 0.77 CYP3A4 (0.37) MAPK1CYP3A4TSHRCD44ALDH1A1
SCHEMBL21317778 0.75 CYP3A4 (0.41) MAPK1CYP3A4TSHRCD44ALDH1A1
SCHEMBL23041366 0.74 CD44 (0.48) MAPK1CYP3A4TSHRCD44ALDH1A1
SCHEMBL25648747 0.73 GRIA1 (0.40) MAPK1CYP3A4TSHRCD44ALDH1A1
SCHEMBL30476125 0.72 CYP3A4 (0.60) MAPK1CYP3A4TSHRCD44ALDH1A1
SCHEMBL272781 0.72 CYP3A4 (0.60) MAPK1CYP3A4TSHRCD44ALDH1A1
SCHEMBL24899747 0.71 CYP3A4 (0.52) MAPK1CYP3A4TSHRCD44ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008076048-A1 INDAZOLYL ESTER AND AMIDE DERIVATIVES FOR THE TREATMENT OF GLUCOCORTICOID RECEPTOR MEDIATED DISORDERS ASTRAZENECA AB (SE) 2008-06-26 WO disclosed