SCHEMBL14189293

SCHEMBL14189293

Cc1ncnc2ccc(-c3ccccc3)cc12

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 8/20 0.65
LMNA P02545 4/20 0.49
BRAF P15056 3/20 0.49
RAF1 P04049 2/20 0.49
PIK3CA P42336 2/20 0.49
PIK3CD O00329 1/20 0.49
PIK3CB P42338 1/20 0.49
MTOR P42345 1/20 0.49
PIK3CG P48736 1/20 0.49
CYP1A2 P05177 5/20 0.48
CYP3A4 P08684 5/20 0.48
CLK4 Q9HAZ1 5/20 0.48
ALDH1A1 P00352 3/20 0.48
USP2 O75604 2/20 0.48
IRAK4 Q9NWZ3 1/20 0.48
MAPK1 P28482 3/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
HSD17B10 Q99714 2/20 0.47
TP53 P04637 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22744963 0.87 MAP4K4 (0.51) MAP4K4LMNACYP1A2CYP3A4CLK4
SCHEMBL14216189 0.84 LMNA (0.46) MAP4K4LMNACYP1A2CYP3A4CLK4
SCHEMBL14189299 0.84 MAP4K4 (0.66) MAP4K4LMNABRAFRAF1PIK3CA
SCHEMBL14189305 0.83 MAP4K4 (0.68) MAP4K4LMNABRAFRAF1CLK4
SCHEMBL14189294 0.81 LMNA (0.44) MAP4K4LMNACYP1A2CYP3A4CLK4
SCHEMBL14189300 0.81 MAP4K4 (0.70) MAP4K4LMNABRAFRAF1PIK3CA
SCHEMBL14189297 0.81 LMNA (0.44) MAP4K4LMNACYP1A2CYP3A4CLK4
SCHEMBL14189303 0.81 CYP1A2 (0.72) LMNABRAFRAF1CYP1A2CYP3A4
SCHEMBL14189296 0.81 MAP4K4 (0.50) MAP4K4LMNACYP1A2CYP3A4CLK4
SCHEMBL14189298 0.81 MAP4K4 (0.72) MAP4K4LMNABRAFRAF1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7378409-B2 Substituted cycloalkylamine derivatives as modulators of chemokine receptor activity BRISTOL-MYERS SQUIBB COMPANY (US) 2008-05-27 US disclosed
US-7378409-B2 Substituted cycloalkylamine derivatives as modulators of chemokine receptor activity BRISTOL-MYERS SQUIBB COMPANY (US) 2008-05-27 US disclosed