SCHEMBL14192196

SCHEMBL14192196

CCc1nn(C)c2nc(Cl)ncc12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 6/20 0.37
NR3C1 P04150 3/20 0.36
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
GAA P10253 2/20 0.33
PDE4B Q07343 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C19 P33261 1/20 0.32
LRRK2 Q5S007 2/20 0.32
MAPK8 P45983 1/20 0.32
MAPK9 P45984 1/20 0.32
MAPK10 P53779 1/20 0.32
KHK P50053 1/20 0.31
JUN P05412 1/20 0.31
NFKB1 P19838 1/20 0.31
NFKB2 Q00653 1/20 0.31
RELA Q04206 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31729367 0.83 PDE2A (0.35) PDE2ANR3C1KMT2AMEN1GAA
SCHEMBL8089905 0.77 PDE2A (0.40) PDE2ANR3C1KMT2AGAASMN1; SMN2
SCHEMBL2546778 0.76 KHK (0.54) NR3C1KMT2AMEN1GAAKHK
SCHEMBL30259549 0.76 PDE2A (0.39) PDE2AKMT2AGAACYP1A2CYP3A4
SCHEMBL26527418 0.76 PDE2A (0.39) PDE2AKMT2AGAACYP1A2CYP3A4
SCHEMBL30968152 0.76 PDE2A (0.39) PDE2ANR3C1KMT2AGAACYP1A2
SCHEMBL31729399 0.75 PDE2A (0.36) PDE2AKMT2AMEN1GAA
SCHEMBL31728695 0.73 CSNK1A1 (0.39) PDE2AKMT2AGAASMN1; SMN2
SCHEMBL22745727 0.72 PDE4D (0.45) LRRK2
SCHEMBL31729103 0.72 PDE2A (0.36) PDE2AKMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008069997-A1 SUBSTITUTED DIAZEPAN COMPOUNDS AS OREXIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2008-06-12 WO disclosed