SCHEMBL14196147

SCHEMBL14196147

CN(C(=O)OC(C)(C)C)[C@H]1CCN(c2ccc(-n3ccc(CCc4ccccc4)cc3=O)cn2)C1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 7/20 0.50
AAK1 Q2M2I8 2/20 0.45
PDE10A Q9Y233 1/20 0.45
CHRM4 P08173 3/20 0.44
DPP4 P27487 3/20 0.44
RET P07949 2/20 0.40
KCNH2 Q12809 2/20 0.39
DPP8 Q6V1X1 2/20 0.39
DPP9 Q86TI2 2/20 0.39
NAPEPLD Q6IQ20 1/20 0.39
NPC1 O15118 2/20 0.38
ALDH1A1 P00352 2/20 0.38
MAPT P10636 2/20 0.38
RAB9A P51151 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
KDM4E B2RXH2 1/20 0.38
TP53 P04637 1/20 0.38
HPGD P15428 1/20 0.38
HTT P42858 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4891076 0.89 MCHR1 (0.55) MCHR1CHRM4DPP4KCNH2DPP8
SCHEMBL14196136 0.89 MCHR1 (0.66) MCHR1AAK1PDE10ACHRM4DPP4
SCHEMBL14196138 0.89 MCHR1 (0.66) MCHR1AAK1PDE10ACHRM4DPP4
SCHEMBL4877707 0.82 MCHR1 (0.46) MCHR1AAK1PDE10ACHRM4DPP4
SCHEMBL14196144 0.80 MCHR1 (0.64) MCHR1DPP4KCNH2DPP8DPP9
SCHEMBL4888566 0.79 MCHR1 (0.73) MCHR1DPP4KCNH2DPP8DPP9
SCHEMBL4732127 0.79 MCHR1 (0.73) MCHR1DPP4KCNH2DPP8DPP9
SCHEMBL4877733 0.78 MCHR1 (0.71) MCHR1DPP4KCNH2DPP8DPP9
SCHEMBL1782082 0.76 MCHR1 (0.49) MCHR1DPP4
SCHEMBL4732287 0.75 MCHR1 (0.51) MCHR1CHRM4DPP4KCNH2DPP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080085884-A1 Melanin Concentrating Hormone Receptor-1 Antagonist Pyridinones PFIZER INC 2008-04-10 US disclosed
US-20080085884-A1 Melanin Concentrating Hormone Receptor-1 Antagonist Pyridinones PFIZER INC 2008-04-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080085884-A1 Melanin Concentrating Hormone Receptor-1 Antagonist Pyridinones MCHR1, MCHR2, MC1R MCHR1 1/4885AAK1 888/4885PDE10A 683/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.