SCHEMBL14199037

SCHEMBL14199037

CN(C)C(=O)C(=O)c1cn(CC=O)c2ccccc12

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
CNR2 P34972 1/20 0.47
KMT2A Q03164 2/20 0.47
ADORA1 P30542 2/20 0.46
NR4A2 P43354 1/20 0.45
HDAC1 Q13547 2/20 0.44
HDAC6 Q9UBN7 2/20 0.44
HDAC2 Q92769 1/20 0.44
CREBBP Q92793 1/20 0.44
L3MBTL1 Q9Y468 2/20 0.43
KDM4E B2RXH2 1/20 0.43
GAA P10253 1/20 0.43
KAT2B Q92831 1/20 0.42
MAPK1 P28482 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23927841 0.85 CNR2 (0.65) ALDH1A1SMN1; SMN2CNR2KMT2AADORA1
SCHEMBL19232823 0.81 CREBBP (0.64) ALDH1A1SMN1; SMN2KMT2ACREBBPL3MBTL1
SCHEMBL3242026 0.78 ALDH1A1 (0.58) ALDH1A1SMN1; SMN2KMT2ANR4A2
SCHEMBL19234284 0.77 PTPN7 (0.61) ALDH1A1SMN1; SMN2CNR2KMT2ANR4A2
SCHEMBL19234287 0.77 KMT2A (0.51) ALDH1A1CNR2KMT2AADORA1NR4A2
SCHEMBL19233876 0.74 KDM4E (0.70) ALDH1A1SMN1; SMN2CNR2KMT2ANR4A2
SCHEMBL8527697 0.71 MEN1 (0.55) ALDH1A1SMN1; SMN2KMT2AHDAC1HDAC6
SCHEMBL1538812 0.69 NR4A2 (0.66) ALDH1A1SMN1; SMN2KMT2AADORA1NR4A2
SCHEMBL15155216 0.69 KAT2B (0.65) ALDH1A1SMN1; SMN2KMT2ACREBBPL3MBTL1
SCHEMBL7778088 0.69 CNR2 (0.70) ALDH1A1SMN1; SMN2CNR2KMT2ACREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1608627-B1 BICYCLIC ANILIDE SPIROHYDANTOIN CGRP RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2008-05-07 EP disclosed
US-7202251-B2 Bicyclic anilide spirohydantoin CGRP receptor antagonists MERCK & CO., INC. (US) 2007-04-10 US disclosed
US-7202251-B2 Bicyclic anilide spirohydantoin CGRP receptor antagonists MERCK & CO., INC. (US) 2007-04-10 US disclosed