SCHEMBL14200033

SCHEMBL14200033

COBN(C)C1CCN(CCC2CCOc3cc(S(=O)(=O)c4cccc(F)c4)ccc32)C1

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.40
HTR2A P28223 3/20 0.38
HTR2C P28335 1/20 0.38
HTR6 P50406 14/20 0.37
HTR1A P08908 2/20 0.37
DRD2 P14416 2/20 0.37
HTR7 P34969 2/20 0.37
PKM P14618 1/20 0.36
PKLR P30613 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2957622 0.89 HTR2A (0.42) KCNH2HTR2AHTR2CHTR6HTR1A
SCHEMBL13240503 0.85 HTR2A (0.39) KCNH2HTR2AHTR2CHTR6HTR1A
SCHEMBL2953292 0.84 HTR2A (0.39) KCNH2HTR2AHTR2CHTR6HTR1A
SCHEMBL2952107 0.81 HTR6 (0.40) KCNH2HTR2AHTR6HTR1ADRD2
SCHEMBL2952104 0.80 HTR6 (0.47) KCNH2HTR2AHTR6DRD2HTR7
Hydrochloric Acid SCHEMBL2963663 0.80 HTR6 (0.46) KCNH2HTR2AHTR6DRD2HTR7
SCHEMBL2963683 0.73 HTR6 (0.49) HTR6PKMPKLR
SCHEMBL2953919 0.73 HTR6 (0.44) HTR6PKMPKLR
SCHEMBL2953515 0.71 HTR6 (0.48) HTR6PKMPKLR
SCHEMBL2960638 0.71 HTR6 (0.53) HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1831191-B1 CHROMAN DERIVATIVES AND THEIR USE AS 5-HT RECEPTOR LIGANDS HOFFMANN LA ROCHE (CH) 2008-05-21 EP disclosed