SCHEMBL14200823

SCHEMBL14200823

CCCC(C)N(C(=O)CC(C)(C)C)c1cc(C)ccc1F

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 7/20 0.34
PSEN2 P49810 7/20 0.34
APH1B Q8WW43 7/20 0.34
NCSTN Q92542 7/20 0.34
APH1A Q96BI3 7/20 0.34
PSENEN Q9NZ42 7/20 0.34
AKR1B1 P15121 1/20 0.33
TAS1R3 Q7RTX0 1/20 0.33
TAS1R1 Q7RTX1 1/20 0.33
UBE2M P61081 2/20 0.32
DCUN1D1 Q96GG9 2/20 0.32
MAPK14 Q16539 1/20 0.32
RIPK1 Q13546 2/20 0.32
HPGD P15428 2/20 0.32
ALDH1A1 P00352 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
NPC1 O15118 1/20 0.31
MAPT P10636 1/20 0.31
PKM P14618 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14201089 0.92 PDE5A (0.35) AKR1B1UBE2MDCUN1D1MAPK14RIPK1
SCHEMBL14200977 0.90 AKR1B1 (0.34) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL14200974 0.89 AKR1B1 (0.34) AKR1B1TAS1R3TAS1R1UBE2MDCUN1D1
SCHEMBL14543478 0.86 PSEN1 (0.36) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL14200825 0.84 POLB (0.33) AKR1B1RIPK1HPGDALDH1A1MEN1
SCHEMBL14201091 0.84 AKR1B1 (0.35) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL14201197 0.83 PSEN1 (0.34) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL14200779 0.81 PSEN1 (0.32) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL14229315 0.80 PSEN1 (0.35) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL14201018 0.80 PSEN1 (0.33) PSEN1PSEN2APH1BNCSTNAPH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed