SCHEMBL14201089

SCHEMBL14201089

CCCCCC(C)N(C(=O)CC(C)(C)C)c1cc(C)ccc1F

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 1/20 0.35
MLYCD O95822 1/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
ALDH1A1 P00352 1/20 0.33
TP53 P04637 1/20 0.33
GPX4 P36969 1/20 0.33
PAX8 Q06710 1/20 0.33
POLB P06746 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
MAPT P10636 1/20 0.32
PKM P14618 1/20 0.32
AKR1B1 P15121 1/20 0.32
UBE2M P61081 1/20 0.31
DCUN1D1 Q96GG9 1/20 0.31
MAPK14 Q16539 1/20 0.31
CNR1 P21554 1/20 0.30
CNR2 P34972 1/20 0.30
RIPK1 Q13546 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14200823 0.92 PSEN1 (0.34) NPC1RAB9AALDH1A1SMN1; SMN2MAPT
SCHEMBL14228981 0.87 PDE5A (0.35) PDE5AMLYCDNPC1RAB9AALDH1A1
SCHEMBL14200977 0.87 AKR1B1 (0.34) NPC1RAB9ASMN1; SMN2MAPTPKM
SCHEMBL14200825 0.86 POLB (0.33) PDE5ANPC1RAB9AALDH1A1TP53
SCHEMBL14201198 0.84 PDE5A (0.33) PDE5AMLYCDNPC1RAB9AALDH1A1
SCHEMBL14200974 0.83 AKR1B1 (0.34) NPC1RAB9AALDH1A1SMN1; SMN2MAPT
SCHEMBL14200885 0.82
SCHEMBL14229434 0.81 PDE5A (0.34) PDE5AMLYCDNPC1RAB9AALDH1A1
SCHEMBL14200872 0.81 MLYCD (0.33) MLYCD
SCHEMBL14201091 0.81 AKR1B1 (0.35) NPC1RAB9ASMN1; SMN2MAPTPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed