SCHEMBL14201573

SCHEMBL14201573

CCCC(CCC)S(=O)(=O)CC(C)C(=O)N[C@@H](Cc1cc(F)cc(F)c1)[C@H](O)CNCc1cccc(CC)c1

nearest known ligand 0.79

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.79
CTSB P07858 19/20 0.79
CTSD P07339 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5645966 0.91 BACE1 (0.78) BACE1CTSBCTSD
SCHEMBL14348040 0.91 BACE1 (0.78) BACE1CTSBCTSD
SCHEMBL14348042 0.91 BACE1 (0.78) BACE1CTSBCTSD
SCHEMBL14347930 0.90 CTSB (0.84) BACE1CTSB
Hydrochloric Acid SCHEMBL4666330 0.90 BACE1 (0.76) BACE1CTSBCTSD
Hydrochloric Acid SCHEMBL6708069 0.90 CTSB (0.83) BACE1CTSB
SCHEMBL6685299 0.90 CTSB (0.85) BACE1CTSB
SCHEMBL14347932 0.90 CTSB (0.85) BACE1CTSB
SCHEMBL14201300 0.90 CTSB (0.75) BACE1CTSB
SCHEMBL14347931 0.89 CTSB (0.84) BACE1CTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1395551-B1 HYDROXY ALKYL AMINE DERIVATIVES AS BETA-SECRETASE INHIBITORS AND THEIR USE FOR THE TREATMENT OF ALZHEIMER'S DISEASE AND SIMILAR DISEASES ELAN PHARM INC (US) 2008-05-21 EP disclosed