SCHEMBL14205481

SCHEMBL14205481

CCCCN1CCN(CCCOc2ccc3nc(-c4ccc(OCCc5ccc(Cl)cc5)cc4)n(CCCC)c3c2)CC1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.49
AGER Q15109 5/20 0.49
HRH4 Q9H3N8 1/20 0.47
HRH2 P25021 2/20 0.46
HRH1 P35367 2/20 0.46
DRD2 P14416 5/20 0.46
DRD3 P35462 5/20 0.46
ESR1 P03372 1/20 0.45
HRH3 Q9Y5N1 3/20 0.45
ADRA1A P35348 2/20 0.45
KCNH2 Q12809 2/20 0.45
CXCR1 P25024 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1283067 0.97 AGER (0.53) MAPTAGERHRH4HRH2HRH1
SCHEMBL1283065 0.97 AGER (0.49) MAPTAGERHRH4HRH2HRH1
SCHEMBL1283792 0.96 AGER (0.51) MAPTAGERDRD2DRD3ESR1
SCHEMBL1283563 0.94 MAPT (0.46) MAPTAGERHRH4HRH2HRH1
SCHEMBL1283170 0.94 AGER (0.52) MAPTAGERHRH4DRD2DRD3
SCHEMBL1283281 0.93 ESR1 (0.54) MAPTAGERDRD2DRD3ESR1
SCHEMBL1283809 0.93 ESR1 (0.54) MAPTAGERDRD2DRD3ESR1
SCHEMBL1282811 0.91 ESR1 (0.45) MAPTAGERHRH4HRH2HRH1
SCHEMBL1282993 0.91 ESR1 (0.46) MAPTAGERDRD2DRD3ESR1
SCHEMBL1283432 0.91 BRD4 (0.50) MAPTAGERESR1HRH3ADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7361678-B2 Azole derivatives and fused bicyclic azole derivatives as therapeutic agents TRANSTECH PHARMA, INC. (US) 2008-04-22 US disclosed
US-7361678-B2 Azole derivatives and fused bicyclic azole derivatives as therapeutic agents TRANSTECH PHARMA, INC. (US) 2008-04-22 US disclosed