SCHEMBL14212434

SCHEMBL14212434

O=c1n(Cc2ccc(C(F)(F)F)nc2)nc2c(-c3ccc(F)cc3)c(-c3ccc(Cl)cc3)cnn12

nearest known ligand 0.85

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 15/20 0.85
CYP2C9 P11712 5/20 0.53
CYP2C19 P33261 5/20 0.53
CYP3A4 P08684 4/20 0.53
MEN1 O00255 2/20 0.40
RAB9A P51151 2/20 0.40
KMT2A Q03164 2/20 0.40
NPC1 O15118 1/20 0.40
NR3C1 P04150 1/20 0.40
NR1H2 P55055 1/20 0.38
NR1H3 Q13133 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14211892 0.96 CNR1 (0.91) CNR1CYP2C9CYP2C19CYP3A4NR3C1
SCHEMBL14211170 0.94 CNR1 (0.86) CNR1CYP2C9CYP2C19CYP3A4NR3C1
SCHEMBL14211173 0.93 CNR1 (0.85) CNR1CYP2C9CYP2C19CYP3A4MEN1
SCHEMBL14181112 0.93 CNR1 (0.85) CNR1CYP2C9CYP2C19CYP3A4NR3C1
SCHEMBL4798385 0.92 CNR1 (1.00) CNR1CYP2C9CYP2C19CYP3A4RAB9A
SCHEMBL14212433 0.92 CNR1 (0.84) CNR1CYP2C9CYP2C19CYP3A4NR3C1
SCHEMBL14212187 0.92 CNR1 (0.84) CNR1CYP2C9CYP2C19CYP3A4NR3C1
SCHEMBL14181114 0.91 CNR1 (0.79) CNR1CYP2C9CYP2C19CYP3A4NR3C1
SCHEMBL14212429 0.91 CNR1 (0.79) CNR1CYP2C9CYP2C19CYP3A4NR3C1
SCHEMBL14211878 0.91 CNR1 (0.79) CNR1CYP2C9CYP2C19CYP3A4NR3C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7378418-B2 Azabicyclic heterocycles as cannabinoid receptor modulators BRISTOL-MYERS SQUIBB COMPANY (US) 2008-05-27 US disclosed
EP-1697370-B1 AZABICYCLIC HETEROCYCLES AS CANNABINOID RECEPTOR MODULATORS BRISTOL MYERS SQUIBB CO (US) 2007-04-25 EP disclosed