SCHEMBL14216880

SCHEMBL14216880

C=Nc1cc(OCCCN2CCOCC2)c(OC)cc1C#N

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 7/20 0.52
CYP2D6 P10635 1/20 0.51
TSHR P16473 1/20 0.51
SRC P12931 9/20 0.51
ABL1 P00519 3/20 0.50
BCR P11274 2/20 0.50
RAF1 P04049 1/20 0.49
MAPK3 P27361 1/20 0.49
MAPK1 P28482 1/20 0.49
FYN P06241 1/20 0.49
EGFR P00533 2/20 0.48
ERBB2 P04626 1/20 0.48
CHEK1 O14757 1/20 0.48
FLT1 P17948 1/20 0.47
KDR P35968 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14421313 0.86 MAP2K1 (0.52) MAP2K1CYP2D6TSHRSRCABL1
SCHEMBL5027821 0.85 MAP2K1 (0.49) MAP2K1CYP2D6TSHRSRCABL1
SCHEMBL5027818 0.85 MAP2K1 (0.49) MAP2K1CYP2D6TSHRSRCABL1
SCHEMBL17922753 0.85 MAP2K1 (0.49) MAP2K1CYP2D6TSHRSRCABL1
SCHEMBL2163402 0.83 MAP2K1 (0.55) MAP2K1CYP2D6TSHRSRCABL1
SCHEMBL3281444 0.83 MAP2K1 (0.55) MAP2K1CYP2D6TSHRSRCABL1
Hydrochloric Acid SCHEMBL27950647 0.82 MAP2K1 (0.54) MAP2K1CYP2D6TSHRSRCABL1
SCHEMBL14421398 0.79 CYP2D6 (0.56) MAP2K1CYP2D6TSHRSRCABL1
SCHEMBL3280339 0.79 CYP2D6 (0.56) MAP2K1CYP2D6TSHRSRCABL1
SCHEMBL5023805 0.77 LMNA (0.54) MAP2K1CYP2D6SRCABL1BCR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1299381-B1 SUBSTITUTED QUINAZOLINE DERIVATIVES AND THEIR USE AS INHIBITORS ASTRAZENECA AB (SE) 2008-05-07 EP disclosed