SCHEMBL14217522

SCHEMBL14217522

COc1ccc(COc2ccc(-c3noc(CC(NC(=O)OC(C)(C)C)C(=O)O)n3)nc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 3/20 0.48
PPARG P37231 2/20 0.48
PTPN1 P18031 4/20 0.47
ITGB3 P05106 1/20 0.44
ITGA2B P08514 1/20 0.44
ITGA4 P13612 2/20 0.42
ITGB7 P26010 2/20 0.42
BCL2 P10415 1/20 0.42
ALDH1A1 P00352 1/20 0.41
CACNA1B Q00975 1/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
PRSS1 P07477 1/20 0.40
PRSS2 P07478 1/20 0.40
PRSS3 P35030 1/20 0.40
TPSAB1 Q15661 1/20 0.40
TPH1 P17752 2/20 0.40
FFAR1 O14842 1/20 0.40
HCAR2 Q8TDS4 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14217521 0.89 CACNA1B (0.41) PPARAPPARGPTPN1ITGB3ITGA2B
SCHEMBL13250886 0.86 HCAR2 (0.49) PTPN1ITGB3ITGA2BHCAR2CYP2C9
SCHEMBL13225536 0.83 PTPN1 (0.43) PTPN1ALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL14217523 0.83 PTPN1 (0.38) PPARAPPARGPTPN1BCL2ALDH1A1
SCHEMBL4548463 0.82 CYP4F2 (0.53) ALDH1A1NPC1RAB9ASMN1; SMN2FFAR1
SCHEMBL4548432 0.82 HCAR2 (0.49) PTPN1ALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL13933857 0.78 NPC1 (0.41) PTPN1ALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL4548429 0.76 MAOB (0.46) ALDH1A1NPC1RAB9ASMN1; SMN2TPH1
SCHEMBL4548407 0.75 LMNA (0.52) ALDH1A1NPC1RAB9ASMN1; SMN2FFAR1
SCHEMBL13933915 0.75 HCAR2 (0.48) HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008051403-A2 NIACIN RECEPTOR AGONISTS, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF TREATMENT MERCK & CO., INC. (US) 2008-05-02 WO disclosed