SCHEMBL14219639

SCHEMBL14219639

Bc1cnc(Nc2c(C(=O)NOCCO)ccc(F)c2F)c(C)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 17/20 0.56
MAP2K2 P36507 4/20 0.55
PIM1 P11309 1/20 0.46
CAMK2B Q13554 1/20 0.46
ABCB11 O95342 1/20 0.42
NQO2 P16083 1/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
CYP3A4 P08684 1/20 0.42
HDAC3 O15379 2/20 0.42
HDAC4 P56524 2/20 0.42
HDAC1 Q13547 2/20 0.42
HDAC7 Q8WUI4 2/20 0.42
HDAC2 Q92769 2/20 0.42
HDAC10 Q969S8 2/20 0.42
HDAC11 Q96DB2 2/20 0.42
HDAC8 Q9BY41 2/20 0.42
HDAC6 Q9UBN7 2/20 0.42
HDAC9 Q9UKV0 2/20 0.42
HDAC5 Q9UQL6 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14219611 0.89 MAP2K1 (0.62) MAP2K1MAP2K2PIM1CAMK2BABCB11
SCHEMBL14219652 0.89 MAP2K1 (0.43) MAP2K1MAP2K2ABCB11NQO2
SCHEMBL14220152 0.88 MAP2K1 (0.63) MAP2K1MAP2K2PIM1CAMK2BABCB11
SCHEMBL14219641 0.86 MAP2K1 (0.54) MAP2K1MAP2K2PIM1CAMK2BMAPK1
SCHEMBL14219653 0.82 MAP2K1 (0.60) MAP2K1MAP2K2PIM1CAMK2BABCB11
SCHEMBL4596340 0.81 MAP2K1 (0.64) MAP2K1MAP2K2PIM1CAMK2BCYP2C9
SCHEMBL14220178 0.79 MAP2K1 (0.41) MAP2K1MAP2K2ABCB11NQO2
SCHEMBL14220160 0.79 MAP2K1 (0.49) MAP2K1MAP2K2ABCB11NQO2
SCHEMBL14220150 0.79 MAP2K1 (0.48) MAP2K1MAP2K2PIM1CAMK2BHDAC3
SCHEMBL14223208 0.79 MEN1 (0.43) MAP2K1MAP2K2PIM1CAMK2BABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1908751-A1 N-hydroxy benzamides with antitumour activity EOS S.p.A. (IT) 2008-04-09 EP disclosed