SCHEMBL14229346

SCHEMBL14229346

CCCCN(CCC)S(=O)(=O)N(C)c1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.48
TDP1 Q9NUW8 1/20 0.46
CA1 P00915 2/20 0.44
NR1I2 O75469 1/20 0.41
RAB9A P51151 2/20 0.40
ESR2 Q92731 1/20 0.40
NPC1 O15118 1/20 0.40
JAK2 O60674 1/20 0.40
PAX8 Q06710 1/20 0.40
CA12 O43570 3/20 0.40
CA9 Q16790 3/20 0.40
CA2 P00918 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
SLC22A6 Q4U2R8 1/20 0.40
SLC22A8 Q8TCC7 1/20 0.40
ABCC2 Q92887 1/20 0.40
SLC22A12 Q96S37 1/20 0.40
UGT1A7 Q9HAW7 1/20 0.40
SLC22A11 Q9NSA0 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14200318 0.83 CA1 (0.40) ESR1TDP1CA1RAB9ACA12
SCHEMBL14229111 0.75 CA1 (0.58) ESR1TDP1CA1RAB9AESR2
SCHEMBL14229180 0.74 CA1 (0.79) ESR1TDP1CA1RAB9ACA12
SCHEMBL25137428 0.74 CA12 (0.55) NR1I2CA12CA9CA2SMN1; SMN2
SCHEMBL13762630 0.73 CA12 (0.50) ESR1TDP1CA12CA9CA2
SCHEMBL14229181 0.73 CA1 (0.61) TDP1CA1RAB9ACA12CA9
SCHEMBL8910873 0.73 CA12 (0.43) ESR1TDP1RAB9ANPC1JAK2
Lithium SCHEMBL31041149 0.72 CA12 (0.53) NR1I2CA12CA9CA2SMN1; SMN2
SCHEMBL25137433 0.70 CA12 (0.52) ESR1NR1I2CA12CA9CA2
SCHEMBL2057475 0.70 TDP1 (0.73) ESR1TDP1CA1NR1I2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed