SCHEMBL14229382

SCHEMBL14229382

CCCCN(c1nccc(CCC)n1)C(C)CCC

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.32
DYRK1A Q13627 1/20 0.31
KDM4E B2RXH2 1/20 0.31
LMNA P02545 1/20 0.31
CYP3A4 P08684 1/20 0.31
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14229496 0.94 KCNH2 (0.35) KCNH2DYRK1ALMNA
SCHEMBL14228949 0.93 KCNH2 (0.34) KCNH2DYRK1AKDM4ELMNACYP3A4
SCHEMBL14229183 0.90 KCNH2 (0.33) KCNH2DYRK1AKDM4ELMNACYP3A4
SCHEMBL14229178 0.90 DYRK1A (0.32) DYRK1A
SCHEMBL14229267 0.88 KCNH2 (0.37) KCNH2DYRK1ALMNA
SCHEMBL14229039 0.87 KCNH2 (0.33) KCNH2KDM4ELMNACYP3A4TSHR
SCHEMBL14200633 0.85 ACACB (0.31)
SCHEMBL14229636 0.84 CRHR1 (0.33) KCNH2KDM4ELMNACYP3A4TSHR
SCHEMBL14229718 0.84 KCNH2 (0.36) KCNH2DYRK1ALMNA
SCHEMBL14229171 0.83 DYRK1A (0.31) DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed