SCHEMBL1423398

SCHEMBL1423398

N#Cc1ccccc1C(N)=NO

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.46
LMNA P02545 2/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
TSHR P16473 1/20 0.39
POLB P06746 3/20 0.38
PPIA P62937 1/20 0.38
MAPT P10636 2/20 0.37
ESR2 Q92731 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
HTT P42858 1/20 0.34
GFER P55789 1/20 0.34
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1423395 1.00 GAA (0.46) GAALMNAL3MBTL1TSHRPOLB
SCHEMBL1305313 0.84 TSHR (0.39) GAALMNATSHRPOLBPPIA
SCHEMBL10454257 0.82 TSHR (0.38) GAALMNAL3MBTL1TSHRPOLB
SCHEMBL2995386 0.82 TSHR (0.38) GAALMNAL3MBTL1TSHRPOLB
SCHEMBL9045774 0.80 GAA (0.46) GAALMNAL3MBTL1TSHRMAPT
SCHEMBL1259760 0.76 TSHR (0.39) GAALMNATSHRPOLBPPIA
SCHEMBL1259761 0.76 TSHR (0.39) GAALMNATSHRPOLBPPIA
SCHEMBL262368 0.75 NPC1 (0.58) GAALMNATSHRPOLBPPIA
SCHEMBL11229875 0.75 TSHR (0.41) GAALMNATSHRPOLBPPIA
Bromide SCHEMBL28425575 0.73 NPC1 (0.56) GAALMNATSHRPOLBPPIA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2297140-A1 NOVEL 1,2,4 OXADIAZOLE COMPOUNDS AND METHODS OF USE THEREOF Abbott Laboratories (US) 2011-03-23 EP disclosed
WO-2009148452-A1 NOVEL 1,2,4 OXADIAZOLE COMPOUNDS AND METHODS OF USE THEREOF ABBOTT LABORATORIES (US) 2009-12-10 WO disclosed