SCHEMBL14239134

SCHEMBL14239134

CC1(C)COc2nc3cc(-c4ccccn4)ccc3c(=O)n2C1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.39
CYP3A4 P08684 1/20 0.38
PIK3CD O00329 4/20 0.38
PIK3CA P42336 4/20 0.38
PIK3CG P48736 4/20 0.38
PIK3CB P42338 3/20 0.38
TGFBR1 P36897 1/20 0.36
METAP2 P50579 1/20 0.36
CTSD P07339 1/20 0.36
BACE1 P56817 1/20 0.36
RET P07949 2/20 0.35
RIPK1 Q13546 1/20 0.35
RIPK3 Q9Y572 1/20 0.35
PKMYT1 Q99640 1/20 0.35
DHODH Q02127 1/20 0.34
PRMT5 O14744 2/20 0.34
WDR77 Q9BQA1 1/20 0.34
TNKS O95271 1/20 0.33
CNR2 P34972 1/20 0.33
ALOX5AP P20292 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12059073 0.82 NPC1 (0.40) CYP3A4PIK3CDPIK3CAPIK3CGPIK3CB
SCHEMBL14238838 0.80 POLB (0.44) KMT2A
SCHEMBL6920771 0.80 KDM4E (0.39) CYP3A4PIK3CDPIK3CAPIK3CGPIK3CB
SCHEMBL6922413 0.80 NPC1 (0.43) KMT2ACYP3A4PIK3CDPIK3CAPIK3CG
SCHEMBL6922591 0.80 CYP3A4 (0.41) CYP3A4PIK3CDPIK3CAPIK3CGPIK3CB
SCHEMBL6923262 0.78 RAB9A (0.46) KMT2ACYP3A4
SCHEMBL6921660 0.78 CYP3A4 (0.38) CYP3A4PIK3CDPIK3CAPIK3CGPIK3CB
SCHEMBL15818032 0.78 KMT2A (0.39) KMT2APIK3CDPIK3CAPIK3CGPIK3CB
SCHEMBL14239415 0.78 RAB9A (0.41) CYP3A4PIK3CDPIK3CAPIK3CGPIK3CB
SCHEMBL6921117 0.78 CYP3A4 (0.37) CYP3A4PIK3CDPIK3CAPIK3CGPIK3CB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012170845-A2 METABOTROPIC GLUTAMATE RECEPTOR 5 MODULATORS AND METHODS OF USE THEREOF HEFFERNAN MICHELE L R (US) 2012-12-13 WO disclosed