SCHEMBL14239366

SCHEMBL14239366

c1cnc2c(c1)ccn2OC1CCNCC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.39
IRAK4 Q9NWZ3 2/20 0.39
PARP1 P09874 1/20 0.38
SLC6A4 P31645 2/20 0.36
HTR2C P28335 2/20 0.36
HTR2A P28223 1/20 0.36
HTR1A P08908 2/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A3 Q01959 1/20 0.36
HTR3E A5X5Y0 1/20 0.36
HTR3B O95264 1/20 0.36
HTR3A P46098 1/20 0.36
HTR3D Q70Z44 1/20 0.36
HTR3C Q8WXA8 1/20 0.36
HRH1 P35367 1/20 0.36
CYP2C19 P33261 1/20 0.35
CDC7 O00311 1/20 0.35
CDK2 P24941 1/20 0.35
CHRNB2 P17787 1/20 0.35
CHRNA4 P43681 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21062409 0.75 HRH1 (0.43) SLC6A4HTR2CHTR2AHTR1ASLC6A2
SCHEMBL14239400 0.74 HRH1 (0.44) HTR2CHRH1
SCHEMBL15491855 0.72 DAO (0.42) TP53PARP1SLC6A4SLC6A2HTR3A
SCHEMBL4589677 0.71 PARP1 (0.46) TP53PARP1CYP2C19CDC7CDK2
Hydrochloric Acid SCHEMBL14645490 0.70 HRH1 (0.38) SLC6A4HTR2CHTR2AHTR1ASLC6A2
Hydrochloric Acid SCHEMBL27800371 0.67 HTR2C (0.46) PARP1SLC6A4HTR2CHTR2AHTR1A
SCHEMBL14239490 0.66 NR1H4 (0.46) TP53SLC6A4HTR1ASLC6A2SLC6A3
SCHEMBL22689265 0.66 PARP1 (0.45) PARP1SLC6A4CYP2C19CDC7CDK2
SCHEMBL4063072 0.66 HTR6 (0.51)
SCHEMBL3715640 0.66 DDB1 (0.53) TP53SLC6A4HTR2CHTR2AHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012169649-A1 INDAZOLE- AND PYRROLOPYRIDINE-DERIVATIVE AND PHARMACEUTICAL USE THEREOF DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2012-12-13 WO disclosed