SCHEMBL14239807

SCHEMBL14239807

CC(C)(O)C1Cc2nc3cc(-c4ccccn4)ccc3c(=O)n2C1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
CYP3A4 P08684 1/20 0.37
NSD2 O96028 1/20 0.36
TGFBR1 P36897 1/20 0.35
METAP2 P50579 2/20 0.35
DHODH Q02127 1/20 0.35
ABL1 P00519 2/20 0.35
BCR P11274 1/20 0.35
RET P07949 2/20 0.34
RIPK1 Q13546 1/20 0.34
RIPK3 Q9Y572 1/20 0.34
PDK1 Q15118 1/20 0.34
PDK2 Q15119 1/20 0.34
PKMYT1 Q99640 1/20 0.34
MAPT P10636 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
GSK3B P49841 1/20 0.34
DYRK1A Q13627 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14238860 0.90 METAP2 (0.38) NPC1RAB9ATDP1CYP3A4NSD2
SCHEMBL14240292 0.88 CYP3A4 (0.36) NPC1RAB9ATDP1CYP3A4NSD2
SCHEMBL14238851 0.88 METAP2 (0.39) NPC1RAB9ATDP1CYP3A4NSD2
SCHEMBL6920430 0.84 CYP3A4 (0.40) NPC1RAB9ATDP1CYP3A4NSD2
SCHEMBL6921685 0.82 NPC1 (0.39) NPC1RAB9ATDP1CYP3A4NSD2
SCHEMBL14239974 0.81 POLB (0.42) NPC1RAB9ATDP1NSD2ABL1
SCHEMBL14238846 0.80 NPC1 (0.41) NPC1RAB9ATDP1CYP3A4NSD2
SCHEMBL14238847 0.80 CYP3A4 (0.38) NPC1RAB9ATDP1CYP3A4NSD2
SCHEMBL14240294 0.80 USP30 (0.37) NPC1RAB9ATDP1CYP3A4NSD2
SCHEMBL12059330 0.79 CYP3A4 (0.39) NPC1RAB9ATDP1CYP3A4TGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012170845-A2 METABOTROPIC GLUTAMATE RECEPTOR 5 MODULATORS AND METHODS OF USE THEREOF HEFFERNAN MICHELE L R (US) 2012-12-13 WO disclosed