SCHEMBL1424855

SCHEMBL1424855

CC(=O)N1CCN(C(=O)Nc2ccc(F)cc2)CC1

nearest known ligand 0.71

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.71
SMN1; SMN2 Q16637 2/20 0.67
ALDH1A1 P00352 3/20 0.66
POLB P06746 2/20 0.66
CA12 O43570 2/20 0.62
CA1 P00915 2/20 0.62
CA2 P00918 2/20 0.62
CA9 Q16790 2/20 0.62
MAPT P10636 2/20 0.60
PANK3 Q9H999 1/20 0.60
GLA P06280 1/20 0.60
CYP2D6 P10635 1/20 0.57
MEN1 O00255 1/20 0.57
FAAH O00519 1/20 0.56
NPC1 O15118 1/20 0.55
RAB9A P51151 1/20 0.55
NAMPT P43490 1/20 0.55
LMNA P02545 1/20 0.54
HTT P42858 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10053027 0.87 KMT2A (0.71) KMT2ASMN1; SMN2ALDH1A1POLBCA12
SCHEMBL22218903 0.85 KMT2A (0.73) KMT2ASMN1; SMN2ALDH1A1POLBCA12
SCHEMBL4508859 0.84 KMT2A (0.90) KMT2ASMN1; SMN2ALDH1A1POLBCA12
SCHEMBL6538815 0.84 KMT2A (0.67) KMT2ASMN1; SMN2ALDH1A1POLBCA12
SCHEMBL14590776 0.83 LMNA (0.66) KMT2ASMN1; SMN2ALDH1A1CA12CA2
SCHEMBL28956323 0.83 KMT2A (0.61) KMT2ASMN1; SMN2ALDH1A1POLBCA12
SCHEMBL491293 0.83 KMT2A (1.00) KMT2ASMN1; SMN2ALDH1A1CA12CA1
SCHEMBL14590550 0.83 KDM4E (0.71) KMT2AALDH1A1POLBMAPTGLA
SCHEMBL20236278 0.83 KMT2A (0.65) KMT2ASMN1; SMN2ALDH1A1POLBCA12
SCHEMBL10244956 0.83 KMT2A (0.65) KMT2ASMN1; SMN2ALDH1A1POLBCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140836-B1 AMIDE COMPOUNDS ASTELLAS PHARMA INC (JP) 2011-03-23 EP disclosed
US-20040092528-A1 Agent for modulating excitatory synaptic transmission comprising a compound having alpha7 nicotinic acetylcholine receptor activation property FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-05-13 US disclosed
US-6710043-B1 POSSESS THE POTENTIATION OF THE CHOLINERGIC ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2004-03-23 US disclosed
US-20040014745-A1 Amide compounds FUJISAWA PHARMACEUTICAL CO. LTD. (JP) 2004-01-22 US disclosed
EP-1315494-A1 AGENT FOR MODULATING EXCITATORY SYNAPTIC TRANSMISSION COMPRISING A COMPOUND HAVING ALPHA-7 NICOTINIC ACETYLCHOLINE RECEPTOR ACTIVATION PROPERTY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-06-04 EP disclosed
EP-1235575-A2 AGENT FOR EXPRESSION OF LONG-TERM POTENTIATION OF SYNAPTIC TRANSMISSION COMPRISING COMPOUND HAVING BRAIN SOMATOSTATIN ACTIVATION PROPERTY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-09-04 EP disclosed
WO-2002020016-A1 AGENT FOR MODULATING EXCITATORY SYNAPTIC TRANSMISSION COMPRISING A COMPOUND HAVING ALPHA α7 NICOTINIC ACETYLCHOLINE RECEPTOR ACTIVATION PROPERTY FUJISAWA PHARMACEUTICAL CO, LTD (JP) 2002-03-14 WO disclosed
WO-2000072834-A9 AGENT FOR EXPRESSION OF LONG-TERM POTENTIATION OF SYNAPTIC TRANSMISSION COMPRISING COMPOUND HAVING BRAIN SOMATOSTATIN ACTIVATION PROPERTY FUJISAWA PHARMACEUTICAL CO (JP) 2001-12-20 WO disclosed
EP-1140836-A1 AMIDE COMPOUNDS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-10-10 EP disclosed
WO-2000072834-A2 AGENT FOR EXPRESSION OF LONG-TERM POTENTIATION OF SYNAPTIC TRANSMISSION COMPRISING COMPOUND HAVING BRAIN SOMATOSTATIN ACTIVATION PROPERTY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-12-07 WO disclosed
WO-2000042011-A1 AMIDE COMPOUNDS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-07-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040014745-A1 Amide compounds CHRM1, CHRM2, CHRNE KMT2A 1224/4885SMN1; SMN2 1339/4885ALDH1A1 1088/4885
US-20040092528-A1 Agent for modulating excitatory synaptic transmission comprising a compound having alpha7 nicotinic acetylcholine receptor activation property CHRNA7, CHRNA5, CHRNA10 KMT2A 4093/4885SMN1; SMN2 622/4885ALDH1A1 2011/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.