SCHEMBL14249258

SCHEMBL14249258

FC(F)(F)Oc1ccc(-c2nc(Cl)nc3c2ncn3C2CCCCO2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
YTHDC1 Q96MU7 1/20 0.54
TEAD1 P28347 2/20 0.41
TEAD4 Q15561 2/20 0.41
TEAD2 Q15562 2/20 0.41
TEAD3 Q99594 2/20 0.41
CYP2C19 P33261 1/20 0.41
CYP1A2 P05177 1/20 0.40
TSHR P16473 1/20 0.40
TP53 P04637 1/20 0.38
CYP2C9 P11712 1/20 0.38
NFKB1 P19838 1/20 0.38
MAPK1 P28482 1/20 0.38
HSD17B10 Q99714 1/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
APEX1 P27695 1/20 0.38
PI4KA P42356 1/20 0.38
BLM P54132 1/20 0.38
KMT2A Q03164 1/20 0.38
ADCY1 Q08828 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14250027 0.87 YTHDC1 (0.60) YTHDC1CYP2C19CYP1A2TSHRTP53
SCHEMBL14249352 0.87 YTHDC1 (0.57) YTHDC1CYP2C19CYP1A2TSHRTP53
SCHEMBL14248883 0.86 YTHDC1 (0.60) YTHDC1CYP2C19CYP1A2TSHRTP53
SCHEMBL3025868 0.84 YTHDC1 (0.60) YTHDC1CYP2C19CYP1A2TSHRTP53
SCHEMBL3029027 0.84 YTHDC1 (0.60) YTHDC1CYP2C19CYP1A2TSHRTP53
SCHEMBL13765749 0.84 YTHDC1 (0.62) YTHDC1CYP2C19CYP1A2TSHRTP53
SCHEMBL14296940 0.81 YTHDC1 (0.60) YTHDC1CYP2C19CYP1A2TSHRTP53
SCHEMBL3016722 0.81 YTHDC1 (0.57) YTHDC1CYP2C19CYP1A2TSHRTP53
SCHEMBL14249516 0.81 YTHDC1 (0.57) YTHDC1CYP2C19CYP1A2TSHRTP53
SCHEMBL14249905 0.81 MERTK (0.44) YTHDC1TEAD1TEAD4TEAD2TEAD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012172043-A1 PURINE DERIVATIVES AND THEIR USE AS PHARMACEUTICALS FOR PREVENTION OR TREATMENT OF BACTERIAL INFECTIONS LABORATOIRE BIODIM (FR) 2012-12-20 WO disclosed
WO-2012172043-A1 PURINE DERIVATIVES AND THEIR USE AS PHARMACEUTICALS FOR PREVENTION OR TREATMENT OF BACTERIAL INFECTIONS LABORATOIRE BIODIM (FR) 2012-12-20 WO disclosed