SCHEMBL14267653

SCHEMBL14267653

Cc1onc(-c2ccc(S(C)(=O)=O)cc2)c1-c1ccccc1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 17/20 0.77
PTGS1 P23219 4/20 0.77
MT-CO2 P00403 3/20 0.77
CA12 O43570 1/20 0.77
CA1 P00915 1/20 0.77
CA2 P00918 1/20 0.77
LMNA P02545 1/20 0.77
CA3 P07451 1/20 0.77
ADRB2 P07550 1/20 0.77
ADRB1 P08588 1/20 0.77
CYP3A4 P08684 1/20 0.77
ADORA3 P0DMS8 1/20 0.77
CHRM1 P11229 1/20 0.77
ADRA2B P18089 1/20 0.77
CA4 P22748 1/20 0.77
CA6 P23280 1/20 0.77
SLC6A2 P23975 1/20 0.77
PDE4A P27815 1/20 0.77
ADORA1 P30542 1/20 0.77
CA5A P35218 1/20 0.77

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5703656 1.00 PTGS2 (0.77) PTGS2PTGS1MT-CO2CA12CA1
SCHEMBL7474889 0.91 PTGS2 (0.65) PTGS2PTGS1MT-CO2CA12CA1
SCHEMBL28961699 0.90 PTGS2 (0.79) PTGS2PTGS1MT-CO2CA12CA1
SCHEMBL6171081 0.90 PTGS2 (0.79) PTGS2PTGS1MT-CO2CA12CA1
SCHEMBL5422595 0.88 PTGS2 (0.77) PTGS2PTGS1MT-CO2CA12CA1
Valdecoxib SCHEMBL3356 0.87 PTGS2 (1.00) PTGS2PTGS1MT-CO2CA12CA1
SCHEMBL6167941 0.87 PTGS2 (1.00) PTGS2PTGS1MT-CO2CA12CA1
SCHEMBL6168344 0.87 PTGS2 (1.00) PTGS2PTGS1MT-CO2CA12CA1
SCHEMBL6013897 0.87 PTGS2 (0.76) PTGS2PTGS1MT-CO2CA12CA1
SCHEMBL6262268 0.87 PTGS2 (0.75) PTGS2PTGS1MT-CO2CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220106275-A1 RADIOLABELED COMPOUNDS AND USES THEREOF THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK 2022-04-07 US disclosed
WO-2020257653-A1 RADIOLABELED COMPOUNDS AND USES THEREOF THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2020-12-24 WO disclosed
US-7329401-B2 Cyclooxygenase-2 selective agents useful as imaging probes and related methods THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2008-02-12 US disclosed
US-20070286801-A1 CYCLOOXYGENASE-2 SELECTIVE AGENTS USEFUL AS IMAGING PROBES AND RELATED METHODS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2007-12-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070286801-A1 CYCLOOXYGENASE-2 SELECTIVE AGENTS USEFUL AS IMAGING PROBES AND RELATED METHODS PTGS2, PTGES2, PTGER2 PTGS2 1/4885PTGS1 4/4885MT-CO2 520/4885
US-20220106275-A1 RADIOLABELED COMPOUNDS AND USES THEREOF PAICS, TMEM14C, SLCO1B1 PTGS2 4365/4885PTGS1 3758/4885MT-CO2 3290/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.