SCHEMBL14286141

SCHEMBL14286141

O=C(Nc1nc2ccccc2[nH]1)c1cc(-n2cncc2-c2cccc(F)c2F)c[nH]1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 11/20 0.47
PKM P14618 5/20 0.47
TP53 P04637 2/20 0.47
LMNA P02545 2/20 0.47
GAA P10253 1/20 0.47
RAB9A P51151 10/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
KDM4E B2RXH2 1/20 0.45
HSD17B10 Q99714 1/20 0.45
MAOB P27338 1/20 0.43
ADORA2A P29274 1/20 0.43
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
POLB P06746 1/20 0.42
CASP3 P42574 1/20 0.42
SENP8 Q96LD8 1/20 0.42
SENP7 Q9BQF6 1/20 0.42
SENP6 Q9GZR1 1/20 0.42
MTOR P42345 2/20 0.41
IRAK4 Q9NWZ3 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14286131 0.86 POLB (0.52) LMNAGAARAB9ASMN1; SMN2KDM4E
SCHEMBL10067396 0.84 NPC1 (0.48) NPC1PKMTP53LMNAGAA
SCHEMBL5036482 0.79 CYP2C9 (0.35) IRAK4
SCHEMBL14286130 0.78 MAPK14 (0.40)
SCHEMBL14600759 0.72 POLB (0.52) LMNAGAARAB9ASMN1; SMN2KDM4E
SCHEMBL14286150 0.71 GSK3B (0.51) NPC1LMNAGAARAB9AKDM4E
SCHEMBL11706898 0.66 NPC1 (1.00) NPC1PKMTP53LMNAGAA
SCHEMBL14286143 0.66 MAPK1 (0.46) NPC1TP53RAB9ASMN1; SMN2MEN1
SCHEMBL11703736 0.64 NPC1 (0.91) NPC1PKMTP53RAB9ASMN1; SMN2
SCHEMBL28376644 0.64 NPC1 (1.00) NPC1PKMTP53LMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7314885-B2 Pyrrole compounds useful as kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-01-01 US disclosed
US-7314885-B2 Pyrrole compounds useful as kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-01-01 US disclosed