SCHEMBL14287594

SCHEMBL14287594

COc1cccc2c1CN(C(=O)OC(C)(C)C)CC2

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABHD6 Q9BV23 3/20 0.55
ESR2 Q92731 1/20 0.53
NR1H2 P55055 1/20 0.52
MAPK1 P28482 1/20 0.49
MAPT P10636 2/20 0.47
KDM4E B2RXH2 1/20 0.47
DRD2 P14416 1/20 0.46
DRD1 P21728 1/20 0.46
DRD5 P21918 1/20 0.46
DRD3 P35462 1/20 0.46
MTNR1A P48039 1/20 0.45
MTNR1B P49286 1/20 0.45
DDB1 Q16531 1/20 0.45
CRBN Q96SW2 1/20 0.45
P2RX3 P56373 1/20 0.45
MKNK1 Q9BUB5 1/20 0.45
NOTUM Q6P988 1/20 0.45
PTGDR2 Q9Y5Y4 1/20 0.45
GRM5 P41594 1/20 0.44
GRM1 Q13255 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16637999 0.88 ABHD6 (0.65) ABHD6ESR2NR1H2MAPK1MTNR1A
SCHEMBL15062790 0.88 ESR2 (0.51) ABHD6ESR2NR1H2MAPK1MAPT
SCHEMBL21659367 0.86 ESR2 (0.47) ABHD6ESR2NR1H2MAPK1MAPT
SCHEMBL19608875 0.85 ESR2 (0.56) ABHD6ESR2NR1H2MAPK1MAPT
SCHEMBL16518212 0.85 ABHD6 (0.46) ABHD6ESR2NR1H2MAPK1PTGDR2
SCHEMBL16268884 0.84 PTGDR2 (0.52) ABHD6ESR2NR1H2MAPK1DDB1
SCHEMBL30199091 0.84 ESR2 (0.59) ABHD6ESR2NR1H2MAPK1MAPT
SCHEMBL3693657 0.84 ESR2 (0.59) ABHD6ESR2NR1H2MAPK1MAPT
SCHEMBL19178532 0.83 ESR2 (0.47) ABHD6ESR2NR1H2MAPK1DDB1
SCHEMBL4519564 0.83 NR1H2 (0.60) ABHD6ESR2NR1H2MAPK1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7314937-B2 Non-imidazole aryl alkylamines compounds as histamine H3 receptor antagonists, preparation and therapeutic uses ELI LILLY AND COMPANY (US) 2008-01-01 US disclosed
US-7314937-B2 Non-imidazole aryl alkylamines compounds as histamine H3 receptor antagonists, preparation and therapeutic uses ELI LILLY AND COMPANY (US) 2008-01-01 US disclosed