SCHEMBL14292829

SCHEMBL14292829

Cc1cc(C#N)cc(C(=O)c2c(C(C)C)c(=O)[nH]c(=O)n2Cc2cc(N)nc(Cl)n2)c1

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.32
NOS1 P29475 1/20 0.32
NOS2 P35228 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
XDH P47989 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL501833 0.92 KDM4E (0.32) KDM4EALDH1A1HPGD
SCHEMBL14292830 0.89 MEN1 (0.31) MEN1KMT2ATDP1KDM4EALDH1A1
SCHEMBL14292828 0.87 KDM4E (0.33) KDM4EALDH1A1HPGD
SCHEMBL10265355 0.87 KMT2A (0.33) MEN1KMT2ATDP1KDM4EALDH1A1
SCHEMBL10204393 0.85 KMT2A (0.32) NOS3NOS1NOS2MEN1KMT2A
SCHEMBL501684 0.84 MEN1 (0.33) NOS3NOS1NOS2MEN1KMT2A
SCHEMBL10204674 0.83 XDH (0.32) MEN1KMT2ATDP1KDM4EALDH1A1
SCHEMBL10265710 0.82 XDH (0.32) MEN1KMT2ATDP1KDM4EALDH1A1
SCHEMBL10204772 0.82 GRIN1 (0.40)
SCHEMBL10204378 0.82 KDM4E (0.34) MEN1KMT2ATDP1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008016522-A2 HIV REVERSE TRANSCRIPTASE INHIBITORS GILEAD SCIENCES, INC. (US) 2008-02-07 WO disclosed