SCHEMBL14293136

SCHEMBL14293136

COc1cc(OCc2ccccc2)cc(-c2cc(=O)c3ccc(OCC(O)CNC(C)(C)C)cc3o2)c1

nearest known ligand 0.75

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.49
ADRB1 P08588 1/20 0.49
ADRB3 P13945 1/20 0.49
TNKS O95271 1/20 0.47
CYP19A1 P11511 1/20 0.47
ACHE P22303 1/20 0.46
TERT O14746 1/20 0.45
CYP2D6 P10635 1/20 0.44
KDM4E B2RXH2 1/20 0.44
USP2 O75604 1/20 0.44
ALDH1A1 P00352 1/20 0.44
CYP3A4 P08684 1/20 0.44
HPGD P15428 1/20 0.44
MAPK1 P28482 1/20 0.44
RECQL P46063 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HSD17B10 Q99714 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1483979 0.97 ADRB2 (0.52) ADRB2ADRB1ADRB3ACHECYP2D6
SCHEMBL1483981 0.97 ADRB2 (0.52) ADRB2ADRB1ADRB3ACHECYP2D6
SCHEMBL1483974 0.97 ADRB2 (0.52) ADRB2ADRB1ADRB3ACHECYP2D6
SCHEMBL4412877 0.91 CYP3A4 (0.49) TNKSCYP19A1ACHECYP2D6KDM4E
SCHEMBL4407561 0.86 CYP1A1 (0.48) ADRB2ADRB1ADRB3CYP2D6
SCHEMBL1483644 0.85 ADRB2 (0.47) ADRB2ADRB1ADRB3ACHECYP2D6
SCHEMBL1484227 0.85 ADRB2 (0.47) ADRB2ADRB1ADRB3ACHECYP2D6
SCHEMBL1483645 0.85 ADRB2 (0.47) ADRB2ADRB1ADRB3ACHECYP2D6
SCHEMBL1484581 0.85 ABCB1 (0.46)
SCHEMBL4399919 0.83 MEN1 (0.47) TNKSCYP2D6KDM4EALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008018089-A1 R-(-) / S-(+)-7-[3-N-SUBSTITUTED AMINO-2-HYDROXYPROPOXY] FLAVONES COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2008-02-14 WO disclosed