SCHEMBL14293233

SCHEMBL14293233

CC1=NOCC1CNC(=O)OC1CCc2c(sc(NC(=O)CC(C)c3cccnc3)c2N)C1

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
RAB9A P51151 1/20 0.35
KCNA5 P22460 1/20 0.32
MAPT P10636 3/20 0.32
ADORA2B P29275 3/20 0.31
TP53 P04637 1/20 0.31
ADORA2A P29274 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
ADRB3 P13945 2/20 0.31
KCNH2 Q12809 2/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
SLC6A4 P31645 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12895477 0.83 KDM4E (0.35) KDM4EALDH1A1RAB9AKCNA5MAPT
SCHEMBL12895371 0.83 KDM4E (0.35) KDM4EALDH1A1RAB9AKCNA5MAPT
SCHEMBL14292425 0.81 KDM4E (0.38) KDM4EALDH1A1RAB9AMAPTADORA2B
SCHEMBL14292364 0.79 HPGD (0.40) RAB9AMAPTTP53CYP3A4
SCHEMBL12895275 0.78 RAB9A (0.36) KDM4EALDH1A1RAB9AKCNA5MAPT
SCHEMBL14292368 0.78 RAB9A (0.44) KDM4EALDH1A1RAB9AKCNA5MAPT
SCHEMBL14293248 0.76 KDM4E (0.36) KDM4EALDH1A1RAB9AKCNA5MAPT
SCHEMBL14292979 0.76 HPGD (0.53) ALDH1A1RAB9AMAPTL3MBTL1CYP3A4
SCHEMBL14293234 0.76 HPGD (0.36) KDM4EALDH1A1RAB9AMAPTTP53
SCHEMBL14292397 0.76 HPGD (0.37) RAB9AMAPTTP53L3MBTL1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008020045-A1 TETRAHYDROBENZOTHIOPHENE DERIVATIVES 4SC AG (DE) 2008-02-21 WO disclosed