SCHEMBL14293442

SCHEMBL14293442

O=Nc1cc(O)ccc1-c1nnc(O)n1-c1cccc2ccc(F)cc12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 4/20 0.35
IDO2 Q6ZQW0 4/20 0.35
TRPV1 Q8NER1 1/20 0.34
HTR5A P47898 1/20 0.33
HSP90AA1 P07900 2/20 0.32
IDO1 P14902 3/20 0.32
MEN1 O00255 3/20 0.32
RAB9A P51151 3/20 0.32
KMT2A Q03164 3/20 0.32
KDM4E B2RXH2 1/20 0.32
MAPT P10636 1/20 0.32
DHODH Q02127 2/20 0.32
NPC1 O15118 2/20 0.31
APAF1 O14727 1/20 0.31
MITF O75030 1/20 0.31
CYP17A1 P05093 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP11B1 P15538 1/20 0.31
CYP11B2 P19099 1/20 0.31
HTR1A P08908 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8931041 0.87 HSP90AA1 (0.40) TDO2IDO2TRPV1HTR5AHSP90AA1
SCHEMBL13808428 0.82 HSP90AA1 (0.39) TDO2IDO2TRPV1HTR5AHSP90AA1
SCHEMBL14345588 0.79 TDO2 (0.42) TDO2IDO2HSP90AA1IDO1MEN1
SCHEMBL2596721 0.78 TDO2 (0.39) TDO2IDO2HSP90AA1IDO1MEN1
SCHEMBL931818 0.74 HSP90AA1 (0.43) HSP90AA1MEN1KMT2ADHODHCYP17A1
SCHEMBL8931043 0.70 HSP90AA1 (0.68) TDO2IDO2HTR5AHSP90AA1KDM4E
SCHEMBL13983092 0.69 HSP90AA1 (0.56) TDO2IDO2HSP90AA1
SCHEMBL4936858 0.67 HSP90AA1 (0.60) HSP90AA1KMT2AKDM4EMAPTL3MBTL1
SCHEMBL930881 0.66 HSP90AA1 (0.50) HSP90AA1KMT2AKDM4EMAPTL3MBTL1
SCHEMBL930856 0.65 HSP90AA1 (0.39) TDO2IDO2HSP90AA1IDO1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008021364-A2 TRIAZOLE COMPOUNDS THAT MODULATE HSP90 ACTIVITY SYNTA PHARMACEUTICALS CORP. (US) 2008-02-21 WO disclosed