SCHEMBL1429675

SCHEMBL1429675

CC1CC2(CCN1)CNS(=O)(=O)N2c1cccc(F)c1

nearest known ligand 0.62

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 18/20 0.62
ALOX5 P09917 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1170550 1.00 BACE1 (0.62) BACE1ALOX5
SCHEMBL1170384 1.00 BACE1 (0.62) BACE1ALOX5
SCHEMBL1170554 0.88 BACE1 (0.48) BACE1
SCHEMBL7716203 0.83 BACE1 (0.43) BACE1ALOX5
SCHEMBL14685963 0.83 BACE1 (0.43) BACE1ALOX5
SCHEMBL1170881 0.81 BACE1 (0.58) BACE1ALOX5
SCHEMBL16494479 0.79 BACE1 (0.69) BACE1
SCHEMBL4318021 0.79 BACE1 (0.69) BACE1
SCHEMBL4307297 0.79 BACE1 (0.69) BACE1
SCHEMBL1171152 0.77 BACE1 (1.00) BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2300484-A1 NOVEL CLASS OF SPIRO PIPERIDINES FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES Pfizer Inc. (US) 2011-03-30 EP disclosed
WO-2009136350-A1 NOVEL CLASS OF SPIRO PIPERIDINES FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES PFIZER INC. (US) 2009-11-12 WO disclosed