SCHEMBL14302001

SCHEMBL14302001

CCN(CC)CCCC(C)Nc1ccn2ncc(Br)c2n1

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CCR4 P51679 4/20 0.49
CACNA2D1 P54289 8/20 0.44
KCNH3 Q9ULD8 1/20 0.41
TMEM97 Q5BJF2 5/20 0.40
SIGMAR1 Q99720 5/20 0.40
SLC2A1 P11166 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4333039 0.81 RET (0.45) CACNA2D1
SCHEMBL14302002 0.78 CCR4 (0.53) CCR4TMEM97SIGMAR1
SCHEMBL14356890 0.78 CCR4 (0.50) CCR4TMEM97SIGMAR1
SCHEMBL13122757 0.73 GSK3B (0.64)
SCHEMBL23148336 0.72 NTRK1 (0.43)
SCHEMBL23148335 0.72 NTRK1 (0.43)
SCHEMBL4333275 0.72 AXL (0.33)
SCHEMBL15393779 0.72 GSK3B (0.44) CCR4TMEM97SIGMAR1
SCHEMBL1440944 0.72 CDK2 (0.39)
SCHEMBL1442100 0.72 PIM1 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1873157-A1 Pyrazolopyrimidines and salts thereof, pharmaceutical compositions comprising same, methods of preparing same and uses of same Bayer Schering Pharma Aktiengesellschaft (DE) 2008-01-02 EP disclosed
WO-2007147647-A1 PYRAZOLOPYRIMIDINES AND SALTS THEREOF, PHARMACEUTICAL COMPOSITIONS COMPRISING SAME, METHODS OF PREPARING SAME AND USES OF SAME. BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2007-12-27 WO disclosed