SCHEMBL14304584

SCHEMBL14304584

CCc1cn(C(=O)OC(C)(C)C)c2ccc(OC)cc12

nearest known ligand 0.61

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 11/20 0.61
AKR1C2 P52895 5/20 0.56
HTR6 P50406 2/20 0.55
MTNR1A P48039 5/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
PTGS1 P23219 2/20 0.48
AKR1C4 P17516 1/20 0.48
PDE10A Q9Y233 1/20 0.47
MTNR1B P49286 4/20 0.46
NQO2 P16083 1/20 0.44
AR P10275 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16727061 0.91 AKR1C3 (0.57) AKR1C3AKR1C2HTR6MTNR1AL3MBTL1
SCHEMBL16727064 0.90 AKR1C3 (0.56) AKR1C3AKR1C2HTR6MTNR1AL3MBTL1
SCHEMBL29169601 0.89 HTR6 (0.57) AKR1C3AKR1C2HTR6MTNR1AL3MBTL1
SCHEMBL24723630 0.88 AKR1C3 (0.54) AKR1C3AKR1C2HTR6MTNR1AL3MBTL1
SCHEMBL2724803 0.87 AKR1C3 (0.53) AKR1C3AKR1C2HTR6MTNR1AL3MBTL1
SCHEMBL29993260 0.86 AKR1C3 (0.58) AKR1C3AKR1C2HTR6MTNR1AL3MBTL1
SCHEMBL24877860 0.86 HTR6 (0.76) AKR1C3HTR6MTNR1A
SCHEMBL30485883 0.86 HTR6 (0.76) AKR1C3HTR6MTNR1A
SCHEMBL24723812 0.86 AKR1C3 (0.57) AKR1C3AKR1C2HTR6MTNR1AL3MBTL1
SCHEMBL29992497 0.86 AKR1C3 (0.57) AKR1C3AKR1C2HTR6MTNR1AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008014249-A2 IMPROVED PREPARATIONS OF 2 -SUBSTITUTED PYRROLO [2, 3-B] PYRAZINE ( 4, 7 -DIAZAINDOLE ) COMPOUNDS SANOFI-AVENTIS (FR) 2008-01-31 WO disclosed