SCHEMBL14307499

SCHEMBL14307499

Cc1ccc(Nc2c(F)cccc2Cl)c(CC(=O)Oc2ccc(N=C=S)cc2)c1

nearest known ligand 0.63

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 9/20 0.63
PTGS1 P23219 3/20 0.63
ABCB11 O95342 1/20 0.63
PPARG P37231 1/20 0.63
NR1I3 Q14994 1/20 0.63
CAMK2A Q9UQM7 1/20 0.39
LMNA P02545 2/20 0.37
USP2 O75604 1/20 0.37
TTR P02766 1/20 0.37
CYP2C9 P11712 1/20 0.37
TBXA2R P21731 1/20 0.37
MAPK1 P28482 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15267404 0.92 PTGS2 (0.62) PTGS2PTGS1ABCB11PPARGNR1I3
SCHEMBL15267399 0.85 PTGS2 (0.65) PTGS2PTGS1ABCB11PPARGNR1I3
SCHEMBL2880887 0.84 PTGS2 (0.64) PTGS2PTGS1ABCB11PPARGNR1I3
SCHEMBL2886958 0.84 PTGS2 (0.66) PTGS2PTGS1ABCB11PPARGNR1I3
SCHEMBL5534966 0.82 PTGS2 (0.79) PTGS2PTGS1ABCB11PPARGNR1I3
SCHEMBL2885873 0.81 TTR (0.56) PTGS2PTGS1ABCB11NR1I3CAMK2A
SCHEMBL2888394 0.81 PTGS2 (0.60) PTGS2PTGS1ABCB11PPARGNR1I3
SCHEMBL13688513 0.80 PTGS2 (0.66) PTGS2PTGS1ABCB11PPARGNR1I3
SCHEMBL14307498 0.80 PTGS2 (0.61) PTGS2PTGS1ABCB11PPARGNR1I3
SCHEMBL14308724 0.80 PTGS2 (0.58) PTGS2PTGS1ABCB11PPARGNR1I3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8541398-B2 Hydrogen sulfide derivatives of non-steroidal anti-inflammatory drugs ANTIBE THERAPEUTICS INC. (CA) 2013-09-24 US disclosed
WO-2008009127-A1 HYDROGEN SULFIDE DERIVATIVES OF NON-STEROIDAL ANTI-INFLAMMATORY DRUGS ANTIBE THERAPEUTICS INC. (CA) 2008-01-24 WO disclosed