SCHEMBL143250

SCHEMBL143250

COc1ccc2c(c1)cc1n2-c2ccccc2C1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIK1 P39086 1/20 0.46
GRIK2 Q13002 1/20 0.46
L3MBTL1 Q9Y468 2/20 0.45
POLB P06746 1/20 0.45
HTR6 P50406 1/20 0.45
MAPT P10636 3/20 0.42
NPC1 O15118 1/20 0.42
MAPK1 P28482 1/20 0.42
RAB9A P51151 1/20 0.42
SCN2A Q99250 1/20 0.42
CYP1A2 P05177 1/20 0.41
CYP2A6 P11509 1/20 0.41
TP53 P04637 2/20 0.41
KDM4E B2RXH2 3/20 0.41
ALDH1A1 P00352 3/20 0.41
HPGD P15428 3/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
USP2 O75604 1/20 0.41
TNNI3 P19429 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29930012 1.00 GRIK1 (0.46) GRIK1GRIK2L3MBTL1POLBHTR6
SCHEMBL144090 0.89 MAPT (0.45) L3MBTL1POLBHTR6MAPTNPC1
SCHEMBL29930299 0.89 MAPT (0.45) L3MBTL1POLBHTR6MAPTNPC1
SCHEMBL142584 0.82 MAPT (0.46) POLBMAPTNPC1MAPK1RAB9A
SCHEMBL140833 0.81 MAPT (0.45) L3MBTL1MAPTNPC1MAPK1RAB9A
SCHEMBL29930121 0.81 MAPT (0.45) L3MBTL1MAPTNPC1MAPK1RAB9A
SCHEMBL29929810 0.79 MAPT (0.43) MAPTNPC1MAPK1RAB9AKDM4E
SCHEMBL143400 0.79 MAPT (0.43) MAPTNPC1MAPK1RAB9AKDM4E
SCHEMBL199137 0.78 MAPT (0.39) MAPTNPC1MAPK1RAB9AKDM4E
SCHEMBL144099 0.78 TDO2 (0.49) MAPTNPC1MAPK1RAB9ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115043847-B Preparation method of 10H-indolo [1,2-a ] indol-10-one compound 西北师范大学 2023-05-26 CN disclosed
CN-115043847-A Preparation method of 10H-indolo [1,2-a ] indol-10-one compound 西北师范大学 2022-09-13 CN disclosed
US-8940909-B2 Indicator platform BIOSYNTH AG (CH) 2015-01-27 US disclosed
US-8940909-B2 Indicator platform BIOSYNTH AG (CH) 2015-01-27 US disclosed
EP-2427431-B1 NOVEL INDICATOR PLATFORM BIOSYNTH AG (CH) 2013-05-01 EP disclosed
US-20120058503-A1 Novel Indicator Platform BIOSYNTH AG (CH) 2012-03-08 US disclosed
US-20120058503-A1 Novel Indicator Platform BIOSYNTH AG (CH) 2012-03-08 US disclosed
WO-2010128120-A1 NOVEL INDICATOR PLATFORM BIOSYNTH AG (CH) 2010-11-11 WO disclosed