SCHEMBL14340751

SCHEMBL14340751

Nc1nc(Cl)cc(Nc2cc(N)c(Sc3ccncc3)c(Cl)c2)n1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLA1 P09884 1/20 0.53
ROCK2 O75116 6/20 0.53
MAPT P10636 6/20 0.44
POLB P06746 1/20 0.44
GAA P10253 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
KMT2A Q03164 3/20 0.44
OPRK1 P41145 2/20 0.37
MEN1 O00255 2/20 0.36
CYP3A4 P08684 2/20 0.36
NPC1 O15118 2/20 0.36
CYP2C19 P33261 2/20 0.36
RAB9A P51151 2/20 0.36
CYP1A2 P05177 1/20 0.36
AGPAT2 O15120 1/20 0.36
CDC7 O00311 1/20 0.36
CHEK1 O14757 1/20 0.36
AURKA O14965 1/20 0.36
PDPK1 O15530 1/20 0.36
DAPK3 O43293 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5253850 0.94 POLA1 (0.57) POLA1ROCK2MAPTPOLBGAA
SCHEMBL13115515 0.88 ROCK2 (0.53) POLA1ROCK2MAPTPOLBGAA
SCHEMBL3364603 0.84 ROCK2 (0.56) POLA1ROCK2MAPTPOLBGAA
SCHEMBL5256438 0.82 ROCK2 (0.71) POLA1ROCK2MAPTPOLBGAA
SCHEMBL5253438 0.82 ROCK2 (0.61) POLA1ROCK2CYP3A4AGPAT2ROCK1
SCHEMBL10036353 0.82 POLA1 (0.61) POLA1ROCK2MAPTPOLBGAA
SCHEMBL724445 0.78 AGPAT2 (0.58) ROCK2MAPTKMT2AAGPAT2AURKA
SCHEMBL10036354 0.77 ROCK2 (0.68) POLA1ROCK2OPRK1CYP3A4AGPAT2
SCHEMBL10305603 0.77 ROCK2 (0.40) POLA1ROCK2MAPTPOLBGAA
SCHEMBL10036314 0.76 ROCK2 (0.52) ROCK2MAPTKMT2AMEN1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1470122-B1 RHO-KINASE INHIBITORS BAYER PHARMACEUTICALS CORP (US) 2007-12-19 EP disclosed