SCHEMBL14367229

SCHEMBL14367229

C[C@@H](NC(=O)Cc1cc(F)cc(F)c1)C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 1/20 0.48
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
HTT P42858 1/20 0.46
THRA P10827 2/20 0.46
THRB P10828 2/20 0.46
PSEN1 P49768 11/20 0.46
PSEN2 P49810 11/20 0.46
APH1B Q8WW43 11/20 0.46
NCSTN Q92542 11/20 0.46
APH1A Q96BI3 11/20 0.46
PSENEN Q9NZ42 11/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
TDP1 Q9NUW8 1/20 0.44
GSAP A4D1B5 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4106052 1.00 SMYD3 (0.48) SMYD3KDM4EALDH1A1CYP3A4CYP2D6
SCHEMBL3088596 1.00 SMYD3 (0.48) SMYD3KDM4EALDH1A1CYP3A4CYP2D6
SCHEMBL5966991 0.94 PSEN1 (0.47) SMYD3KDM4EALDH1A1CYP3A4CYP2D6
SCHEMBL3343185 0.85 SMYD3 (0.50) SMYD3KDM4EALDH1A1HTTPSEN1
SCHEMBL4111216 0.84 TSHR (0.50) SMYD3HTTPSEN1PSEN2APH1B
SCHEMBL3343337 0.84 TSHR (0.50) SMYD3HTTPSEN1PSEN2APH1B
SCHEMBL3343088 0.84 THRA (0.52) SMYD3KDM4EALDH1A1CYP3A4CYP2D6
SCHEMBL5967316 0.83 PSEN1 (0.47) SMYD3KDM4EALDH1A1CYP3A4CYP2D6
SCHEMBL5967298 0.83 PSEN1 (0.52) SMYD3PSEN1PSEN2APH1BNCSTN
SCHEMBL2819918 0.83 PSEN1 (0.51) SMYD3ALDH1A1PSEN1PSEN2APH1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7294622-B2 Lactams and uses thereof ASTRAZENECA AB (SE) 2007-11-13 US disclosed
US-7294622-B2 Lactams and uses thereof ASTRAZENECA AB (SE) 2007-11-13 US disclosed