SCHEMBL14376293

SCHEMBL14376293

CC(C)C(=O)N1CC2CC1CN2C

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.44
CHRNB2 P17787 1/20 0.40
CHRNA3 P32297 1/20 0.40
CHRNA4 P43681 1/20 0.40
CHRNB3 Q05901 1/20 0.40
CHRNA6 Q15825 1/20 0.40
VNN1 O95497 1/20 0.38
GSK3B P49841 1/20 0.32
DYRK1A Q13627 1/20 0.32
CHRM2 P08172 2/20 0.32
CHRM4 P08173 2/20 0.32
CHRM5 P08912 2/20 0.32
CHRM1 P11229 2/20 0.32
CHRM3 P20309 2/20 0.32
HSD11B1 P28845 2/20 0.31
DPP4 P27487 3/20 0.30
DPP8 Q6V1X1 3/20 0.30
DPP9 Q86TI2 3/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18347997 1.00 PIK3CD (0.44) PIK3CDCHRNB2CHRNA3CHRNA4CHRNB3
SCHEMBL19869628 1.00 PIK3CD (0.44) PIK3CDCHRNB2CHRNA3CHRNA4CHRNB3
SCHEMBL18347996 1.00 PIK3CD (0.44) PIK3CDCHRNB2CHRNA3CHRNA4CHRNB3
SCHEMBL22916981 0.90 PIK3CD (0.52) PIK3CDCHRNB2CHRNA3CHRNA4CHRNB3
SCHEMBL25514814 0.90 PIK3CD (0.52) PIK3CDCHRNB2CHRNA3CHRNA4CHRNB3
SCHEMBL15451852 0.87 VNN1 (0.34) PIK3CDCHRNB2CHRNA3CHRNA4CHRNB3
SCHEMBL18348016 0.85 PIK3CD (0.41) PIK3CDCHRNB2CHRNA3CHRNA4CHRNB3
SCHEMBL23011816 0.82 PIK3CD (0.46) PIK3CDCHRNB2CHRNA3CHRNA4CHRNB3
SCHEMBL21963795 0.82 PIK3CD (0.46) PIK3CDCHRNB2CHRNA3CHRNA4CHRNB3
SCHEMBL21963809 0.82 PIK3CD (0.46) PIK3CDCHRNB2CHRNA3CHRNA4CHRNB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023096995-A1 COMPOSITIONS AND METHODS COMPRISING SUBSTITUTED N-(2-CHLORO-6-METHYLPHENYL)-2-((6-(6-MEMBERED HETEROCYCLOALKYL)-2-METHYLPYRIMIDIN-4-YL)AMINO)THIAZOLE-5-CARBOXAMIDE ANALOGUES ST. JUDE CHILDREN'S RESEARCH HOSPITAL, INC. (US) 2023-06-01 WO disclosed
US-7276520-B2 Bicyclic piperidine derivatives as melanocortin-4 receptor agonists MERCK & CO., INC. (US) 2007-10-02 US disclosed