SCHEMBL14396502

SCHEMBL14396502

Bc1ccccc1C(=O)Nc1ccc(-n2c(C(F)(F)F)nc3cc(OC)ccc32)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 1/20 0.44
CYP3A4 P08684 3/20 0.43
RUVBL1 Q9Y265 1/20 0.42
PTGES O14684 1/20 0.42
NPC1 O15118 4/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
RAB9A P51151 3/20 0.41
POLB P06746 1/20 0.41
GAA P10253 1/20 0.41
CASP3 P42574 1/20 0.41
SENP7 Q9BQF6 1/20 0.41
SENP6 Q9GZR1 1/20 0.41
AHR P35869 1/20 0.41
ACSS2 Q9NR19 1/20 0.40
METAP2 P50579 1/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2093586 0.90 MAPT (0.50) NPC1MEN1KMT2ARAB9AAHR
SCHEMBL2091863 0.89 MAPT (0.47) TACR3CYP3A4NPC1MEN1KMT2A
SCHEMBL2093496 0.89 NPC1 (0.50) TACR3CYP3A4RUVBL1PTGESNPC1
SCHEMBL2093725 0.89 TACR3 (0.44) TACR3CYP3A4RUVBL1PTGESNPC1
SCHEMBL2092860 0.88 KDR (0.48) TACR3CYP3A4RUVBL1NPC1MEN1
SCHEMBL2094162 0.87 RAB9A (0.52) NPC1MEN1KMT2ARAB9APOLB
SCHEMBL2091845 0.86 NPC1 (0.44) TACR3CYP3A4RUVBL1PTGESNPC1
SCHEMBL2092680 0.86 MEN1 (0.51) MEN1KMT2ARAB9APOLBGAA
SCHEMBL2093163 0.86 HDAC8 (0.46) TACR3NPC1MEN1KMT2ARAB9A
SCHEMBL2090594 0.84 RAB9A (0.58) NPC1MEN1KMT2ARAB9APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007112093-A2 BENZIMIDAZOLYL-PYRIDINE COMPOUNDS FOR INFLAMMATION AND IMMUNE-RELATED USES SYNTA PHARMACEUTICALS CORP. (US) 2007-10-04 WO disclosed