SCHEMBL14404663

SCHEMBL14404663

CCCCN1C(=O)[C@@H]([C@H](O)C(C)C)NC(=O)C12CCN(Cc1ccc(Oc3ccc(CO)cc3)nc1)CC2

nearest known ligand 0.73

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 19/20 0.73
CYP3A4 P08684 1/20 0.61
CYP2D6 P10635 2/20 0.58
CYP2C9 P11712 2/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5339773 0.94 CCR5 (0.73) CCR5CYP3A4CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL6010891 0.93 CCR5 (0.73) CCR5CYP3A4CYP2D6CYP2C9
SCHEMBL5344603 0.93 CCR5 (0.81) CCR5CYP3A4CYP2D6CYP2C9
SCHEMBL5344311 0.93 CCR5 (0.81) CCR5CYP3A4CYP2D6CYP2C9
SCHEMBL6012557 0.93 CCR5 (0.81) CCR5CYP3A4CYP2D6CYP2C9
SCHEMBL19677883 0.93 CCR5 (0.81) CCR5CYP3A4CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL6010720 0.93 CCR5 (0.81) CCR5CYP3A4CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL5815825 0.93 CCR5 (0.81) CCR5CYP3A4CYP2D6CYP2C9
SCHEMBL14381243 0.92 CCR5 (0.70) CCR5CYP3A4CYP2D6CYP2C9
SCHEMBL5344289 0.91 CCR5 (0.87) CCR5CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7285552-B2 Drugs containing triazaspiro[5.5]undecane derivatives as the active ingredient ONO PHARMACEUTICALS CO., LTD. (JP) 2007-10-23 US disclosed
US-7262193-B2 Triazaspiro[5.5]undecane derivative and pharmaceutical composition comprising the same as active ingredient ONO PHARMACEUTICAL CO., LTD. (JP) 2007-08-28 US disclosed