SCHEMBL14409673

SCHEMBL14409673

COc1cc2nccc(Oc3ccc(NC(=O)Nc4cc(C)on4)c(Cl)c3)c2cc1O

nearest known ligand 0.89

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 19/20 0.89
PDGFRA P16234 10/20 0.89
FLT1 P17948 4/20 0.89
FLT4 P35916 4/20 0.89
KIT P10721 3/20 0.89
EPHB2 P29323 2/20 0.89
RIPK2 O43353 2/20 0.89
STK10 O94804 2/20 0.89
ABL1 P00519 2/20 0.89
RET P07949 2/20 0.89
PDGFRB P09619 2/20 0.89
BCR P11274 2/20 0.89
FGFR1 P11362 2/20 0.89
SLC6A3 Q01959 2/20 0.89
DDR1 Q08345 2/20 0.89
MAP4K2 Q12851 2/20 0.89
PTK6 Q13882 2/20 0.89
DDR2 Q16832 2/20 0.89
AURKB Q96GD4 2/20 0.89
RIPK3 Q9Y572 2/20 0.89

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15962810 0.97 KDR (0.89) KDRPDGFRAFLT1FLT4KIT
Tivozanib SCHEMBL29354604 0.94 KDR (1.00) KDRPDGFRAFLT1FLT4KIT
Tivozanib SCHEMBL29354238 0.94 KDR (1.00) KDRPDGFRAFLT1FLT4KIT
Tivozanib SCHEMBL172883 0.94 KDR (1.00) KDRPDGFRAFLT1FLT4KIT
Tivozanib SCHEMBL1869882 0.93 KDR (0.98) KDRPDGFRAFLT1FLT4KIT
Tivozanib SCHEMBL30993908 0.93 KDR (0.98) KDRPDGFRAFLT1FLT4KIT
Tivozanib SCHEMBL21174286 0.92 KDR (0.97) KDRPDGFRAFLT1FLT4KIT
Tivozanib SCHEMBL29394095 0.92 KDR (0.97) KDRPDGFRAFLT1FLT4KIT
Tivozanib SCHEMBL5209537 0.91 KDR (0.93) KDRPDGFRAFLT1FLT4KIT
Tivozanib SCHEMBL5214691 0.91 KDR (0.93) KDRPDGFRAFLT1FLT4KIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1559715-B1 N-{2-CHLORO-4-[(6,7-DIMETHOXY-4-QUINOLYL)OXY]PHENYL}-N'-(5-METHYL-3-ISOXAZOLYL)UREA SALT IN CRYSTALLINE FORM KIRIN BREWERY (JP) 2007-09-26 EP disclosed