SCHEMBL14413751

SCHEMBL14413751

COc1cccc(-c2nc(N)nc(Cl)c2N)c1

nearest known ligand 0.64

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 7/20 0.64
ADORA1 P30542 6/20 0.61
ADORA2B P29275 2/20 0.61
PIK3CG P48736 1/20 0.56
MAPT P10636 1/20 0.53
RXFP1 Q9HBX9 1/20 0.53
HRH2 P25021 1/20 0.51
HRH3 Q9Y5N1 1/20 0.51
DPP4 P27487 1/20 0.50
DHPS P49366 1/20 0.46
TP53 P04637 1/20 0.45
HPGD P15428 1/20 0.45
HTT P42858 1/20 0.45
KDM4E B2RXH2 1/20 0.44
KMT2A Q03164 1/20 0.44
IKBKB O14920 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4905916 0.82 ADORA1 (0.77) ADORA2AADORA1ADORA2BMAPTRXFP1
SCHEMBL14413494 0.82 RIPK2 (0.56) ADORA2AADORA1ADORA2BPIK3CGMAPT
SCHEMBL1892740 0.81 ADORA2A (0.59) ADORA2AADORA1HRH2HRH3HPGD
SCHEMBL10367722 0.80 DHPS (0.62) ADORA2AADORA1ADORA2BMAPTDPP4
SCHEMBL7777497 0.80 ADORA2A (0.58) ADORA2AADORA1ADORA2BPIK3CGMAPT
SCHEMBL17544648 0.78 PIK3CG (0.64) ADORA2AADORA1ADORA2BPIK3CGMAPT
SCHEMBL27631918 0.78 PIK3CG (0.64) ADORA2AADORA1ADORA2BPIK3CGMAPT
SCHEMBL26708031 0.77 KDM4E (0.61) ADORA2AADORA1ADORA2BHPGDHTT
SCHEMBL14413002 0.77 DYRK1A (0.51) ADORA2AADORA1KDM4E
SCHEMBL2321715 0.77 ADORA2A (0.81) ADORA2AADORA1ADORA2BPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007098835-A1 AMINO PYRYMIDINE DERIVATIVES MERCK PATENT GMBH (DE) 2007-09-07 WO disclosed