SCHEMBL14419802

SCHEMBL14419802

NC(=O)c1cc(Cl)c(Cl)c2c1CCCCCO2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.39
MAPK8 P45983 1/20 0.36
ALOX15 P16050 2/20 0.35
MAPK1 P28482 2/20 0.35
HSD17B10 Q99714 2/20 0.35
MEN1 O00255 1/20 0.35
IKBKB O14920 1/20 0.35
USP2 O75604 1/20 0.35
ALDH1A1 P00352 1/20 0.35
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35
MAPK10 P53779 1/20 0.35
KMT2A Q03164 1/20 0.35
NNMT P40261 2/20 0.34
HTR3E A5X5Y0 1/20 0.32
HTR3B O95264 1/20 0.32
HTR3A P46098 1/20 0.32
HTR4 Q13639 1/20 0.32
HTR3D Q70Z44 1/20 0.32
HTR3C Q8WXA8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14419919 0.83 SLC5A1 (0.30)
SCHEMBL8294437 0.78 SLC5A2 (0.32)
SCHEMBL14419808 0.74 PARP1 (0.43) PARP1ALOX15MAPK1HSD17B10MEN1
SCHEMBL8296894 0.72
SCHEMBL8296678 0.72 SLC5A1 (0.31)
SCHEMBL8296680 0.72 PARP1 (0.44) PARP1ALOX15MAPK1HSD17B10MEN1
SCHEMBL7333211 0.71 HTR4 (0.46) HTR3EHTR3BHTR3AHTR4HTR3D
SCHEMBL13315461 0.69 SMN1; SMN2 (0.44) MAPK8HSD17B10MEN1ALDH1A1TP53
SCHEMBL5042500 0.69 HTR4 (0.51) PARP1HTR3EHTR3BHTR3AHTR4
SCHEMBL8295684 0.69 MAPK8 (0.43) PARP1MAPK8MEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1638959-B1 5HT -4 -ANTAGONISTIC 4-(AMINOMETHYL)-PIPERIDINE BENZAMIDES JANSSEN PHARMACEUTICA NV (BE) 2007-09-19 EP disclosed