SCHEMBL14420172

SCHEMBL14420172

CC(C)(O)c1ccc2c(c1)/C(=C/CCN1CCC(C(=O)c3ccc(Cl)cc3)CC1)c1cccnc1CO2

nearest known ligand 0.66

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 2/20 0.66
CHRM2 P08172 1/20 0.56
CCR5 P51681 1/20 0.56
LMNA P02545 2/20 0.39
TSHR P16473 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
HTR2A P28223 1/20 0.39
HTR7 P34969 1/20 0.39
HRH1 P35367 4/20 0.39
KCNH2 Q12809 1/20 0.38
TBXA2R P21731 3/20 0.35
ADRA1D P25100 1/20 0.35
ADRA1A P35348 1/20 0.35
ADRA1B P35368 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
TP53 P04637 1/20 0.34
MAPT P10636 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
MGLL Q99685 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL655909 1.00 CCR1 (0.66) CCR1CHRM2CCR5LMNATSHR
SCHEMBL655908 1.00 CCR1 (0.66) CCR1CHRM2CCR5LMNATSHR
SCHEMBL18633828 0.86 CCR1 (0.62) CCR1CHRM2CCR5HRH1ADRA1D
SCHEMBL15478419 0.86 CCR1 (0.62) CCR1CHRM2CCR5HRH1TBXA2R
SCHEMBL656127 0.86 CCR1 (0.62) CCR1CHRM2CCR5HRH1TBXA2R
SCHEMBL655139 0.86 CCR1 (0.63) CCR1CHRM2CCR5HTR2AHRH1
SCHEMBL655115 0.86 CCR1 (0.63) CCR1CHRM2CCR5HTR2AHRH1
SCHEMBL15478327 0.86 CCR1 (0.70) CCR1CHRM2CCR5LMNATSHR
SCHEMBL3836897 0.86 CCR1 (0.60) CCR1CHRM2CCR5HRH1TBXA2R
SCHEMBL3836896 0.86 CCR1 (0.60) CCR1CHRM2CCR5HRH1TBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7271176-B2 Chemokine receptor antagonists and methods of use thereof MILLENNIUM PHARMACEUTICALS, INC. (US) 2007-09-18 US disclosed